SCHEMBL4012317

SCHEMBL4012317

CC(C)(C)OC(=O)NC1CN(c2ncnc3c2c(-c2ccccc2Cl)cn3CC(=O)O)C1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 9/20 0.49
CNR2 P34972 8/20 0.49
PDE2A O00408 3/20 0.45
PDE10A Q9Y233 1/20 0.40
BTK Q06187 2/20 0.39
KMT2A Q03164 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
DRD2 P14416 2/20 0.37
TP53 P04637 2/20 0.37
MAPT P10636 1/20 0.37
DRD3 P35462 1/20 0.37
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13769679 0.91 CNR1 (0.49) CNR1CNR2PDE2APDE10ABTK
SCHEMBL4009217 0.83 PDE2A (0.46) CNR1CNR2PDE2APDE10ABTK
SCHEMBL4013415 0.82 LMNA (0.39) CNR1CNR2PDE2AKMT2ATP53
SCHEMBL4010459 0.82 MAPT (0.41) CNR1CNR2KMT2ATP53MAPT
SCHEMBL4007954 0.82 MAPT (0.40) CNR1CNR2PDE2AKMT2ATP53
Lithium SCHEMBL4007964 0.82 MAPT (0.40) CNR1CNR2PDE2AKMT2ATP53
SCHEMBL4006053 0.78 LMNA (0.47) CNR1CNR2KMT2ATP53MAPT
Lithium Ion SCHEMBL4007958 0.74 MAPT (0.38) CNR1CNR2PDE2APDE10AKMT2A
SCHEMBL13770196 0.74 MAPT (0.44) CNR1CNR2KMT2ATP53MAPT
SCHEMBL13769540 0.74 CNR1 (0.40) CNR1CNR2KMT2ATP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009080682-A1 PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2009-07-02 WO disclosed