SCHEMBL4013740

SCHEMBL4013740

CN1CC2CC1CN(c1cncc(-c3cc(F)ccc3F)c1)C2

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CHRNB4 P30926 6/20 0.46
CHRNA3 P32297 6/20 0.46
CHRNB2 P17787 1/20 0.37
CHRNA4 P43681 1/20 0.37
CYP11B1 P15538 1/20 0.37
CYP11B2 P19099 1/20 0.37
MAPT P10636 2/20 0.35
GSK3B P49841 2/20 0.35
FAAH O00519 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4013764 0.91 CHRNB4 (0.46) CHRNB4CHRNA3CHRNB2CHRNA4FAAH
SCHEMBL4007838 0.89 CHRNB4 (0.44) CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL2961213 0.79 CHRNB4 (0.60) CHRNB4CHRNA3CHRNB2
SCHEMBL4009078 0.78 CHRNB4 (0.54) CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL2958908 0.77 CHRNB4 (0.42) CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL4004006 0.76 CHRNB4 (0.42) CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL4006470 0.74 HRH3 (0.44) CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL2952778 0.70 CHRNB2 (0.46) CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL2960617 0.69 CHRNB2 (0.62) CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL2961155 0.69 CHRNB2 (0.46) CHRNB4CHRNA3CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081246-A2 BICYCLIC DIAMINES AS NICOTINIC RECEPTOR AGONISTS PFIZER INC. (US) 2009-07-02 WO claimed
WO-2009081246-A2 BICYCLIC DIAMINES AS NICOTINIC RECEPTOR AGONISTS PFIZER INC. (US) 2009-07-02 WO disclosed