SCHEMBL4013812

SCHEMBL4013812

CCCc1nc(=O)c(-c2ccc(OC(C)C)nc2)c(CC)n1Cc1ccc(-c2ccccc2C#N)cc1F

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.39
AGTR1 P30556 11/20 0.38
AGTR2 P50052 9/20 0.38
GRIN1 Q05586 1/20 0.37
GRIN2B Q13224 1/20 0.37
S1PR1 P21453 3/20 0.35
CYP2D6 P10635 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4011619 0.89 AGTR1 (0.42) PPARGAGTR1AGTR2
SCHEMBL1889960 0.88 PPARG (0.40) PPARGAGTR1AGTR2GRIN1GRIN2B
SCHEMBL4012714 0.88 PPARG (0.51) PPARGAGTR1AGTR2
SCHEMBL4008828 0.81 AGTR1 (0.42) PPARGAGTR1AGTR2GRIN1GRIN2B
SCHEMBL4010302 0.81 PPARG (0.50) PPARGAGTR1
SCHEMBL4010555 0.81 PPARG (0.38) PPARGAGTR1AGTR2GRIN1GRIN2B
SCHEMBL4019464 0.80 PPARG (0.54) PPARGAGTR1AGTR2
SCHEMBL2842851 0.78 AGTR1 (0.44) PPARGAGTR1AGTR2
SCHEMBL4308395 0.77 PPARG (0.49) PPARG
SCHEMBL4016615 0.77 PPARG (0.54) PPARGAGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074117-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2009-07-01 EP disclosed
WO-2008062905-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-05-29 WO disclosed