SCHEMBL4013862

SCHEMBL4013862

Cc1cnc2c(C(F)(F)F)cccc2c1-c1cccc(Oc2cccc(S(C)(=O)=O)c2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
NR1H3 Q13133 20/20 1.00
NR1H2 P55055 19/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4018768 0.93 NR1H2 (1.00) NR1H3NR1H2
SCHEMBL4015303 0.92 NR1H3 (0.85) NR1H3NR1H2
SCHEMBL4015435 0.91 NR1H3 (1.00) NR1H3NR1H2
SCHEMBL4012266 0.91 NR1H3 (1.00) NR1H3NR1H2
SCHEMBL4015610 0.91 NR1H3 (0.83) NR1H3NR1H2
SCHEMBL4011906 0.91 NR1H3 (0.83) NR1H3NR1H2
SCHEMBL4012454 0.90 NR1H3 (1.00) NR1H3NR1H2
SCHEMBL4015992 0.89 NR1H3 (0.81) NR1H3NR1H2
SCHEMBL4014656 0.89 NR1H3 (1.00) NR1H3NR1H2
SCHEMBL4009739 0.89 NR1H2 (0.80) NR1H3NR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP claimed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO claimed
US-20230338314-A1 METHODS FOR THE TREATMENT OF MYELOID DERIVED SUPPRESSOR CELLS RELATED DISORDERS THE ROCKEFELLER UNIVERSITY (US) 2023-10-26 US disclosed
US-20230338314-A1 METHODS FOR THE TREATMENT OF MYELOID DERIVED SUPPRESSOR CELLS RELATED DISORDERS THE ROCKEFELLER UNIVERSITY (US) 2023-10-26 US disclosed
US-11648220-B2 Methods for the treatment of myeloid derived suppressor cells related disorders THE ROCKEFELLER UNIVERSITY (US) 2023-05-16 US disclosed
US-11648220-B2 Methods for the treatment of myeloid derived suppressor cells related disorders THE ROCKEFELLER UNIVERSITY (US) 2023-05-16 US disclosed
US-20210220306-A1 TREATMENT AND DIAGNOSIS OF MELANOMA THE ROCKEFELLER UNIVERSITY 2021-07-22 US disclosed
US-10945978-B2 Treatment and diagnosis of melanoma THE ROCKEFELLER UNIVERSITY (US) 2021-03-16 US disclosed
US-20200230090-A1 TREATMENT AND DIAGNOSIS OF MELANOMA THE ROCKEFELLER UNIVERSITY (US) 2020-07-23 US disclosed
US-10543183-B2 Treatment and diagnosis of melanoma THE ROCKEFELLER UNIVERSITY (US) 2020-01-28 US disclosed
US-20190029984-A1 METHODS FOR THE TREATMENT OF MYELOID DERIVED SUPPRESSOR CELLS RELATED DISORDERS THE ROCKEFELLER UNIVERSITY (US) 2019-01-31 US disclosed
US-9526710-B2 Treatment and diagnosis of melanoma THE ROCKEFELLER UNIVERSITY (US) 2016-12-27 US disclosed
US-20160331726-A1 TREATMENT AND DIAGNOSIS OF MELANOMA THE ROCKEFELLER UNIVERSITY (US) 2016-11-17 US disclosed
US-20160331726-A1 TREATMENT AND DIAGNOSIS OF MELANOMA THE ROCKEFELLER UNIVERSITY (US) 2016-11-17 US disclosed
US-9399028-B2 Treatment of drug resistant cancer THE ROCKEFELLER UNIVERSITY (US) 2016-07-26 US disclosed
US-9399028-B2 Treatment of drug resistant cancer THE ROCKEFELLER UNIVERSITY (US) 2016-07-26 US disclosed
US-20150073053-A1 TREATMENT OF DRUG RESISTANT CANCER ROCKEFELLER UNIVERSITY (THE) (US) 2015-03-12 US disclosed
US-20150073053-A1 TREATMENT OF DRUG RESISTANT CANCER ROCKEFELLER UNIVERSITY (THE) (US) 2015-03-12 US disclosed
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10543183-B2 Treatment and diagnosis of melanoma EYA3, BRAF, CD99 NR1H3 4400/4885NR1H2 4537/4885
US-10945978-B2 Treatment and diagnosis of melanoma EYA3, BRAF, CD99 NR1H3 4400/4885NR1H2 4537/4885
US-11648220-B2 Methods for the treatment of myeloid derived suppressor cells related disorders NR1H3, NR1H2, MCL1 NR1H3 1/4885NR1H2 2/4885
US-20230338314-A1 METHODS FOR THE TREATMENT OF MYELOID DERIVED SUPPRESSOR CELLS RELATED DISORDERS NR1H3, NR1H2, MCL1 NR1H3 1/4885NR1H2 2/4885
US-20150073053-A1 TREATMENT OF DRUG RESISTANT CANCER ABCC1, TSG101, NTPCR NR1H3 3331/4885NR1H2 3830/4885
US-20210220306-A1 TREATMENT AND DIAGNOSIS OF MELANOMA EYA3, BRAF, CD99 NR1H3 4400/4885NR1H2 4537/4885
US-20190029984-A1 METHODS FOR THE TREATMENT OF MYELOID DERIVED SUPPRESSOR CELLS RELATED DISORDERS NR1H3, NR1H2, MCL1 NR1H3 1/4885NR1H2 2/4885
US-20200230090-A1 TREATMENT AND DIAGNOSIS OF MELANOMA EYA3, BRAF, CD99 NR1H3 4400/4885NR1H2 4537/4885
US-20160331726-A1 TREATMENT AND DIAGNOSIS OF MELANOMA EYA3, BRAF, CD99 NR1H3 4400/4885NR1H2 4537/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.