SCHEMBL4016047

SCHEMBL4016047

CCOC1=NC(C)=C(c2ccc(OC(C)C)cc2)CN1Cc1ccc(-c2ccccc2-c2noc(=O)[nH]2)cc1

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PPARG P37231 9/20 0.45
AGTR1 P30556 2/20 0.45
KCNH2 Q12809 1/20 0.43
AGTR2 P50052 1/20 0.42
ALDH1A1 P00352 1/20 0.41
SLC33A1 O00400 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4016469 0.88 PPARG (0.52) PPARGAGTR1KCNH2SLC33A1
SCHEMBL4016389 0.87 PPARG (0.58) PPARGAGTR1KCNH2
SCHEMBL4010280 0.81 PPARG (0.52) PPARGAGTR1KCNH2SLC33A1
SCHEMBL1890326 0.79 PPARG (0.53) PPARGAGTR1KCNH2AGTR2
SCHEMBL4016049 0.73 PPARG (0.43) PPARGAGTR1KCNH2
SCHEMBL4010601 0.73 AGTR1 (0.45) PPARGAGTR1SLC33A1
SCHEMBL1890861 0.72 PPARG (0.64) PPARGAGTR1KCNH2
SCHEMBL4016515 0.72 SLC33A1 (0.47) PPARGAGTR1SLC33A1
Bromide SCHEMBL1888121 0.72 PPARG (0.63) PPARGAGTR1KCNH2
SCHEMBL1895526 0.72 PPARG (0.63) PPARGAGTR1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009133970-A1 CRYSTALLINE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-05 WO disclosed
EP-2074117-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2009-07-01 EP disclosed
WO-2008062905-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-05-29 WO disclosed