SCHEMBL4016152

SCHEMBL4016152

Cc1ccc2c(N3CCC(NC(=O)O)CC3)nc(Cl)nc2c1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.44
OPRK1 P41145 2/20 0.43
PRKDC P78527 2/20 0.41
EGLN1 Q9GZT9 2/20 0.40
RAD52 P43351 1/20 0.40
RXFP1 Q9HBX9 1/20 0.39
PAK1 Q13153 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL183884 0.93 PRKDC (0.47) HRH4OPRK1PRKDCRAD52KDM4E
SCHEMBL4019288 0.87 CNR1 (0.46) OPRK1
SCHEMBL4012962 0.85 KDM4E (0.46) OPRK1PRKDCKDM4EALDH1A1HPGD
SCHEMBL4012954 0.85 KDM4E (0.46) OPRK1PRKDCKDM4EALDH1A1HPGD
SCHEMBL4013931 0.81 HRH4 (0.50) HRH4RAD52ALDH1A1
SCHEMBL183991 0.81 PDE10A (0.47) PRKDC
SCHEMBL183992 0.81 PDE10A (0.47) PRKDC
SCHEMBL5503125 0.81 HRH4 (0.52) HRH4PAK1ALDH1A1
SCHEMBL1623785 0.80 SMAD3 (0.54) EGLN1KDM4EALDH1A1HSD17B10
Hydrochloric Acid SCHEMBL4012898 0.80 HRH4 (0.51) HRH4PAK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1784393-B1 QUINAZOLINES USEFUL AS MODULATORS OF ION CHANNELS VERTEX PHARMA (US) 2009-07-01 EP disclosed