SCHEMBL4016465

SCHEMBL4016465

O=CC(N1CCN(c2ccc(F)cc2)CC1)n1cc(Cl)c(-c2ccc(Cl)s2)n1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.35
TSHR P16473 1/20 0.35
HSD17B10 Q99714 1/20 0.35
MAPT P10636 5/20 0.34
DRD2 P14416 2/20 0.34
DRD3 P35462 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
LMNA P02545 2/20 0.34
DRD4 P21917 1/20 0.34
POLB P06746 2/20 0.33
TMEM97 Q5BJF2 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
HTT P42858 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
KCNK3 O14649 1/20 0.33
HSP90AA1 P07900 1/20 0.32
CYP3A4 P08684 2/20 0.32
FLT3 P36888 1/20 0.32
CYP1A2 P05177 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27662974 0.84 MAPT (0.34) ALDH1A1TSHRHSD17B10MAPTDRD2
SCHEMBL4020863 0.79 CCR1 (0.44) ALDH1A1MAPTDRD2DRD3TDP1
SCHEMBL27662971 0.79 ALDH1A1 (0.37) ALDH1A1TSHRHSD17B10MAPTDRD2
SCHEMBL2876645 0.75 CCR1 (0.48) ALDH1A1HSD17B10MAPTPOLBHTT
SCHEMBL4459923 0.74 HSP90AA1 (0.40) ALDH1A1MAPTDRD2DRD3TDP1
SCHEMBL6167745 0.70 MEN1 (0.44) ALDH1A1MAPTTDP1LMNAPOLB
SCHEMBL4014716 0.70 GFER (0.40) ALDH1A1TSHRMAPTDRD2DRD3
SCHEMBL4304948 0.69 MAPT (0.37) ALDH1A1TSHRMAPTDRD2DRD3
SCHEMBL4016082 0.69 DRD2 (0.38) ALDH1A1MAPTDRD2DRD3TDP1
SCHEMBL4019239 0.69 MEN1 (0.40) ALDH1A1TSHRMAPTTDP1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1691810-A4 SUBSTITUTED PIPERAZINES CHEMOCENTRYX INC (US) 2009-07-01 EP disclosed
EP-1691810-A1 SUBSTITUTED PIPERAZINES ChemoCentryx Inc (US) 2006-08-23 EP disclosed
WO-2005056015-A1 SUBSTITUTED PIPERAZINES CHEMOCENTRYX, INC. (US) 2005-06-23 WO disclosed