SCHEMBL4017555

SCHEMBL4017555

CCCCC1=C(Cc2ccc(-c3ccccc3-c3noc(=O)[nH]3)cc2)C(=O)[N]C(C)=N1

nearest known ligand 0.52

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PPARG P37231 10/20 0.51
LTB4R2 Q9NPC1 1/20 0.49
SLC33A1 O00400 3/20 0.48
AGTR1 P30556 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4302459 0.76 AGTR1 (0.52) PPARGLTB4R2SLC33A1AGTR1
SCHEMBL4016594 0.75 SLC33A1 (0.54) PPARGSLC33A1AGTR1
SCHEMBL12348839 0.75 SLC33A1 (0.55) PPARGSLC33A1AGTR1
SCHEMBL4011449 0.74 SLC33A1 (0.53) PPARGSLC33A1AGTR1
SCHEMBL13167983 0.74 PPARG (0.51) PPARGLTB4R2SLC33A1
SCHEMBL4012804 0.74 SLC33A1 (0.47) PPARGLTB4R2SLC33A1AGTR1
SCHEMBL12348453 0.74 LTB4R2 (0.58) LTB4R2SLC33A1AGTR1
SCHEMBL4312659 0.73 PPARG (0.47) PPARGLTB4R2SLC33A1AGTR1
SCHEMBL4016688 0.73 PPARG (0.47) PPARGAGTR1
SCHEMBL4447972 0.73 SLC33A1 (0.51) PPARGLTB4R2SLC33A1AGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009133970-A1 CRYSTALLINE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-05 WO disclosed
EP-2074117-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2009-07-01 EP disclosed
WO-2008062905-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-05-29 WO disclosed