SCHEMBL4018145

SCHEMBL4018145

COC(=O)N(Cc1ccccc1)Cc1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.56
ALDH1A1 P00352 3/20 0.55
NPSR1 Q6W5P4 2/20 0.55
NPC1 O15118 1/20 0.53
RAB9A P51151 1/20 0.53
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
TDP1 Q9NUW8 2/20 0.50
ALOX12 P18054 1/20 0.50
HTT P42858 1/20 0.50
GPR55 Q9Y2T6 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
RECQL P46063 1/20 0.50
TSHR P16473 2/20 0.49
REN P00797 1/20 0.49
CA12 O43570 1/20 0.48
CA9 Q16790 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3328358 0.91 LMNA (0.51) LMNAALDH1A1NPSR1NPC1RAB9A
SCHEMBL15762363 0.91 LMNA (0.66) LMNAALDH1A1NPSR1NPC1MEN1
SCHEMBL9574969 0.88 HDAC1 (0.49) LMNAALDH1A1NPSR1NPC1RAB9A
SCHEMBL18154102 0.88 HDAC1 (0.51) LMNAALDH1A1NPSR1NPC1RAB9A
SCHEMBL7517117 0.85 CTSS (0.51) LMNAALDH1A1NPSR1NPC1RAB9A
SCHEMBL2188007 0.85 HDAC6 (0.56) LMNAREN
SCHEMBL11378934 0.84 NPC1 (0.53) LMNAALDH1A1NPSR1NPC1RAB9A
SCHEMBL2188566 0.84 CNR2 (0.55) LMNAALDH1A1REN
SCHEMBL2095210 0.82 NPC1 (0.67) NPC1RAB9AMEN1KMT2ACA12
SCHEMBL18068879 0.81 CETP (0.43) LMNAALDH1A1NPSR1TDP1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074107-A2 TRICYCLIC COMPOUNDS AS MATRIX METALLOPROTEINASE INHIBITORS Wyeth a Corporation of the State of Delaware (US) 2009-07-01 EP disclosed
WO-2008057254-A2 TRICYCLIC COMPOUNDS AS MATRIX METALLOPROTEINASE INHIBITORS WYETH (US) 2008-05-15 WO disclosed