SCHEMBL4020283

SCHEMBL4020283

Cc1cccc(C2[C@@H](C(=O)c3cccc(O)c3)CN(CCN(C)S(C)(=O)=O)C[C@@H]2C(=O)c2cccc(O)c2)c1F

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.34
KIF11 P52732 1/20 0.34
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
OPRM1 P35372 3/20 0.32
OPRD1 P41143 3/20 0.32
KCNH2 Q12809 1/20 0.31
MCHR1 Q99705 1/20 0.31
BCHE P06276 1/20 0.31
KDM2B Q8NHM5 4/20 0.31
HTR7 P34969 1/20 0.31
MGLL Q99685 1/20 0.31
HTR1A P08908 1/20 0.30
DRD2 P14416 1/20 0.30
DRD1 P21728 1/20 0.30
DRD4 P21917 1/20 0.30
DRD5 P21918 1/20 0.30
DRD3 P35462 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4027285 0.90 MEN1 (0.35) KDM1AOPRM1OPRD1KCNH2MCHR1
SCHEMBL4028041 0.89 OPRM1 (0.35) KDM1AKIF11OPRM1OPRD1KCNH2
SCHEMBL13721487 0.89 OPRM1 (0.35) KDM1AKIF11OPRM1OPRD1KCNH2
SCHEMBL4028045 0.89 OPRM1 (0.35) KDM1AKIF11OPRM1OPRD1KCNH2
SCHEMBL4022438 0.88 KDM1A (0.33) KDM1AKIF11GRIN1GRIN2BOPRM1
SCHEMBL4019903 0.88 KDM1A (0.31) KDM1AKCNH2MCHR1
SCHEMBL4772539 0.87 OPRM1 (0.34) KDM1AOPRM1OPRD1KCNH2MCHR1
SCHEMBL4751548 0.87 OPRM1 (0.34) KDM1AOPRM1OPRD1KCNH2MCHR1
SCHEMBL4751549 0.87 OPRM1 (0.34) KDM1AOPRM1OPRD1KCNH2MCHR1
SCHEMBL4027068 0.86 GRIN1 (0.35) KIF11GRIN1GRIN2BOPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7572814-B2 3,5-dibenzoyl-4-phenyl-piperidine anti-cancer compounds CYTOKINETICS, INCORPORATED (US) 2009-08-11 US claimed