SCHEMBL4024203

SCHEMBL4024203

COC(=O)c1c(C(C)Br)cccc1[N+](=O)[O-]

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.51
CYP1A2 P05177 3/20 0.46
TDP1 Q9NUW8 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
MAPT P10636 3/20 0.44
ABCC4 O15439 2/20 0.44
CACNA1F O60840 2/20 0.44
ABCB11 O95342 2/20 0.44
LMNA P02545 2/20 0.44
ADORA3 P0DMS8 2/20 0.44
ADORA2A P29274 2/20 0.44
ADORA1 P30542 2/20 0.44
OPRM1 P35372 2/20 0.44
SCN1A P35498 2/20 0.44
HTR2B P41595 2/20 0.44
CACNA1D Q01668 2/20 0.44
KCNH2 Q12809 2/20 0.44
CACNA1S Q13698 2/20 0.44
CACNA1C Q13936 2/20 0.44
SCN5A Q14524 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11398188 0.83 TDP1 (0.56) ALDH1A1CYP1A2TDP1L3MBTL1MAPT
SCHEMBL5466810 0.80 ALDH1A1 (0.52) ALDH1A1CYP1A2TDP1L3MBTL1MAPT
SCHEMBL4099183 0.79 TDP1 (0.49) ALDH1A1CYP1A2TDP1L3MBTL1MAPT
SCHEMBL283180 0.78 SMN1; SMN2 (0.47) ALDH1A1CYP1A2TDP1L3MBTL1MAPT
SCHEMBL27738198 0.78 ALDH1A1 (0.46) ALDH1A1MAPTLMNATSHRSMN1; SMN2
SCHEMBL27695016 0.78 ALDH1A1 (0.46) ALDH1A1CYP1A2TDP1L3MBTL1MAPT
SCHEMBL15971290 0.77 CA12 (0.67) ALDH1A1CYP1A2TDP1L3MBTL1MAPT
SCHEMBL50994 0.77 TSHR (0.54) ALDH1A1CYP1A2TDP1L3MBTL1MAPT
SCHEMBL10561907 0.77 CA12 (0.47) L3MBTL1MAPTLMNATSHRKDM4E
SCHEMBL283363 0.77 TDP1 (0.68) ALDH1A1CYP1A2TDP1L3MBTL1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102307871-A Isoindolinone and related analogs as sirtuin modulators SIRTRIS PHARMACEUTICALS INC 2012-01-04 CN disclosed
CN-101495450-A Isoindole derivatives useful for treating pain, gastrointestinal diseases and cancer ASTRAZENECA AB (SE) 2009-07-29 CN disclosed
EP-2029535-A1 ISOINDOLE DERIVATIVES USEFUL FOR TREATING PAIN, GASTROINTESTINAL DISEASES AND CANCER AstraZeneca AB (SE) 2009-03-04 EP disclosed
WO-2007139464-A1 ISOINDOLE DERIVATIVES USEFUL FOR TREATING PAIN, GASTROINTESTINAL DISEASES AND CANCER ASTRAZENECA AB (SE) 2007-12-06 WO disclosed