SCHEMBL4024747

SCHEMBL4024747

CN(Cc1nc(-c2ccccc2F)c(Br)s1)C(=O)OC(C)(C)C.COc1cccc(Sc2sc(CN(C)C(=O)OC(C)(C)C)nc2-c2ccccc2F)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 1/20 0.35
GAA P10253 2/20 0.34
MAPT P10636 2/20 0.34
CLK1 P49759 4/20 0.34
DYRK1A Q13627 3/20 0.34
CLK2 P49760 2/20 0.34
CLK4 Q9HAZ1 1/20 0.34
DYRK1B Q9Y463 1/20 0.34
EDNRA P25101 1/20 0.33
DHFR P00374 1/20 0.33
EGFR P00533 1/20 0.33
PDGFRB P09619 1/20 0.33
KDR P35968 1/20 0.33
GLS O94925 2/20 0.33
SOS1 Q07889 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
HSD17B2 P37059 1/20 0.32
HTT P42858 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3649060 0.91 PTGDR2 (0.31) PTGDR2GAAMAPTGLSSOS1
SCHEMBL3649058 0.88 PTGDR2 (0.31) PTGDR2GAAMAPTSOS1
SCHEMBL3649304 0.87 CLK1 (0.35) PTGDR2CLK1DYRK1ACLK2CLK4
SCHEMBL3650616 0.86 HTR2C (0.37) GLSSOS1HTR2CSLC6A4PDK2
SCHEMBL4024754 0.85 PTGDR2 (0.36) PTGDR2GAAMAPTEDNRADHFR
SCHEMBL4131683 0.85 EDNRA (0.40) PTGDR2GAAMAPTCLK1DYRK1A
SCHEMBL3652888 0.84 GLS (0.34) GLSSOS1HTR2CSLC6A4PDK2
SCHEMBL3647074 0.84 GLS (0.34) GLSSOS1HTR2CSLC6A4PDK2
SCHEMBL3652850 0.84 SOS1 (0.39) GLSSOS1HTR2CSLC6A4PDK2
SCHEMBL3646375 0.83 SOS1 (0.30) SOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed