SCHEMBL4024754

SCHEMBL4024754

CC(C)(C)CN(Cc1nc(-c2ccccc2F)c(Br)s1)C(=O)O.COc1cccc(Sc2sc(CN(CC(C)(C)C)C(=O)O)nc2-c2ccccc2F)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 3/20 0.36
EDNRA P25101 1/20 0.35
MAPT P10636 3/20 0.34
GAA P10253 2/20 0.34
DHFR P00374 1/20 0.33
EGFR P00533 1/20 0.33
PDGFRB P09619 1/20 0.33
KDR P35968 1/20 0.33
DHODH Q02127 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
LPAR1 Q92633 1/20 0.32
LPAR5 Q9H1C0 1/20 0.32
TUBB4A P04350 1/20 0.32
TUBB P07437 1/20 0.32
TUBA3C P0DPH7 1/20 0.32
TUBA1B P68363 1/20 0.32
TUBA4A P68366 1/20 0.32
TUBB4B P68371 1/20 0.32
TUBB3 Q13509 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3649062 0.88 PTGDR2 (0.32) PTGDR2EDNRA
SCHEMBL4024747 0.85 PTGDR2 (0.35) PTGDR2EDNRAMAPTGAADHFR
SCHEMBL3650619 0.85 ALDH1A1 (0.32) PTGDR2MAPTGAAALDH1A1SMN1; SMN2
SCHEMBL3652892 0.84 PPARG (0.33)
SCHEMBL3652856 0.83 ALDH1A1 (0.33) PTGDR2MAPTLPAR1LPAR5ALDH1A1
SCHEMBL4131683 0.83 EDNRA (0.40) PTGDR2EDNRAMAPTGAADHFR
SCHEMBL3647079 0.83
SCHEMBL4024750 0.81 GAA (0.35) PTGDR2EDNRAMAPTGAADHFR
SCHEMBL3646377 0.81
SCHEMBL3649060 0.79 PTGDR2 (0.31) PTGDR2MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed