SCHEMBL4025912

SCHEMBL4025912

CN(C(=O)O)c1cccc2cnccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.49
MAPKAPK2 P49137 1/20 0.49
ROCK1 Q13464 3/20 0.46
LMNA P02545 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
SLC22A12 Q96S37 1/20 0.44
TRPV1 Q8NER1 7/20 0.44
SIGMAR1 Q99720 2/20 0.44
KMT2A Q03164 2/20 0.42
ALDH1A1 P00352 1/20 0.42
ROCK2 O75116 1/20 0.42
HTT P42858 2/20 0.41
MEN1 O00255 1/20 0.41
MAPK1 P28482 1/20 0.41
BLM P54132 1/20 0.41
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2359679 0.86 KDM4E (0.47) KDM4EMAPKAPK2ROCK1LMNACYP1A2
SCHEMBL4025954 0.82 KDM4E (0.49) KDM4EMAPKAPK2ROCK1LMNACYP1A2
SCHEMBL1614544 0.80 SIGMAR1 (0.67) SIGMAR1
SCHEMBL11143333 0.80 KDM4E (0.53) KDM4EMAPKAPK2ROCK1LMNACYP1A2
SCHEMBL29666490 0.80 SIGMAR1 (0.67) SIGMAR1
SCHEMBL28304454 0.79 KDM4E (0.46) KDM4EMAPKAPK2ROCK1LMNACYP1A2
SCHEMBL23951754 0.75 SSTR4 (0.41) ROCK1LMNACYP3A4CYP2D6CYP2C9
SCHEMBL23951463 0.75 SSTR4 (0.41) ROCK1LMNACYP3A4CYP2D6CYP2C9
SCHEMBL23951752 0.75 SSTR4 (0.41) ROCK1LMNACYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL23924314 0.74 SSTR4 (0.41) ROCK1LMNACYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1478363-B1 FUSED AZABICYCLIC COMPOUNDS THAT INHIBIT VANILLOID RECEPTOR SUBTYPE 1 (VR1) RECEPTOR ABBOTT LAB (US) 2009-01-14 EP claimed