SCHEMBL4026658

SCHEMBL4026658

N#CCCCn1c2c(c3cc(C(N)=O)ccc31)CCCC2

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.57
SCARB1 Q8WTV0 6/20 0.48
KDM4E B2RXH2 2/20 0.46
ALDH1A1 P00352 1/20 0.46
HDAC1 Q13547 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
RORC P51449 2/20 0.42
HSD17B10 Q99714 2/20 0.42
MEN1 O00255 1/20 0.42
GLA P06280 1/20 0.42
CASP1 P29466 1/20 0.42
CASP7 P55210 1/20 0.42
KMT2A Q03164 1/20 0.42
ACLY P53396 1/20 0.42
PTGDR2 Q9Y5Y4 2/20 0.41
CHRM2 P08172 1/20 0.41
HTR1A P08908 1/20 0.41
CHRM5 P08912 1/20 0.41
ADRA2A P08913 1/20 0.41
DRD2 P14416 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4024245 0.90 FABP4 (0.50) NPC1SCARB1KDM4EALDH1A1HDAC1
SCHEMBL4028396 0.86 SCARB1 (0.66) NPC1SCARB1HDAC1HDAC6RORC
SCHEMBL13746702 0.77 SCARB1 (0.81) NPC1SCARB1HSD17B10
SCHEMBL4027663 0.74 SCARB1 (0.71) NPC1SCARB1HDAC1HDAC6RORC
SCHEMBL4024931 0.73 SCARB1 (0.69) NPC1SCARB1KDM4EALDH1A1HDAC1
SCHEMBL4029504 0.72 SCARB1 (0.68) NPC1SCARB1KDM4EALDH1A1HDAC1
SCHEMBL4030252 0.72 SCARB1 (0.70) NPC1SCARB1KDM4EALDH1A1HDAC1
SCHEMBL27282251 0.72 CA1 (0.61) NPC1KDM4EALDH1A1HDAC1HDAC6
SCHEMBL4028758 0.71 SCARB1 (0.72) NPC1SCARB1HDAC1HDAC6RORC
SCHEMBL10732414 0.71 CHRM2 (0.64) NPC1SCARB1KDM4EALDH1A1HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009103022-A1 DERIVATIVES OF SUBSTITUTED FUSED RING CYCLOINDOLES AND METHODS OF THEIR USE ITHERX PHARMACEUTICALS, INC. (US) 2009-08-20 WO disclosed
WO-2009103022-A1 DERIVATIVES OF SUBSTITUTED FUSED RING CYCLOINDOLES AND METHODS OF THEIR USE ITHERX PHARMACEUTICALS, INC. (US) 2009-08-20 WO disclosed