SCHEMBL4027006

SCHEMBL4027006

O=C(Nc1cc(C(=O)Nc2c(S(=O)(=O)O)cccc2S(=O)(=O)O)cc(C(=O)Nc2c(S(=O)(=O)O)cccc2S(=O)(=O)O)c1)Nc1cc(C(=O)Nc2c(S(=O)(=O)O)cccc2S(=O)(=O)O)cc(C(=O)Nc2c(S(=O)(=O)O)cccc2S(=O)(=O)O)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TIMP3 P35625 6/20 0.60
MEN1 O00255 7/20 0.50
KMT2A Q03164 7/20 0.50
RECQL P46063 4/20 0.50
HSD17B10 Q99714 4/20 0.50
TDP1 Q9NUW8 4/20 0.50
PKM P14618 4/20 0.50
MAPT P10636 4/20 0.50
CYP1A2 P05177 3/20 0.50
BRCA1 P38398 3/20 0.50
P2RX1 P51575 3/20 0.50
LMNA P02545 3/20 0.50
KDM4E B2RXH2 2/20 0.50
POLB P06746 2/20 0.50
CYP3A4 P08684 2/20 0.50
CYP2C9 P11712 2/20 0.50
NFKB1 P19838 2/20 0.50
APEX1 P27695 2/20 0.50
CYP2C19 P33261 2/20 0.50
STAT1 P42224 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21033369 0.79 TIMP3 (0.68) TIMP3MEN1KMT2ARECQLHSD17B10
SCHEMBL1902159 0.75 TIMP3 (1.00) TIMP3MEN1KMT2ARECQLHSD17B10
SCHEMBL31722454 0.74 KMT2A (0.54) TIMP3MEN1KMT2ARECQLHSD17B10
SCHEMBL11342918 0.74 KMT2A (0.54) TIMP3MEN1KMT2ARECQLHSD17B10
SCHEMBL11337777 0.74 TIMP3 (0.54) TIMP3MEN1KMT2ARECQLHSD17B10
SCHEMBL11496644 0.74 TRPV1 (0.55) TIMP3MEN1KMT2ARECQLHSD17B10
SCHEMBL11348122 0.73 KMT2A (0.51) TIMP3MEN1KMT2ARECQLHSD17B10
SCHEMBL11766235 0.73 KMT2A (0.54) TIMP3MEN1KMT2ARECQLHSD17B10
SCHEMBL11766279 0.73 KMT2A (0.56) TIMP3MEN1KMT2ARECQLHSD17B10
SCHEMBL11339069 0.72 KMT2A (0.53) TIMP3MEN1KMT2ARECQLHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049127-A2 N-METHANOCARBA DERIVATIVES TO TREAT CARDIAC DISEASES University of Connecticut (US) 2009-04-22 EP disclosed
WO-2007139775-A2 N-METHANOCARBA DERIVATIVES TO TREAT CARDIAC DISEASES UNIVERSITY OF CONNECTICUT (US) 2007-12-06 WO disclosed