SCHEMBL4028646

SCHEMBL4028646

Cc1cc(C)cc(OCCCCl)c1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.50
ALOX15 P16050 1/20 0.50
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
KDM4E B2RXH2 1/20 0.44
MAPT P10636 1/20 0.44
ALDH1A1 P00352 3/20 0.39
HTT P42858 1/20 0.39
RAB9A P51151 1/20 0.39
LMNA P02545 1/20 0.39
MAOA P21397 1/20 0.39
SLC6A2 P23975 1/20 0.39
CYP3A4 P08684 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
NPC1 O15118 1/20 0.37
DRD2 P14416 1/20 0.37
DRD4 P21917 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL974357 0.86 ALDH1A1 (0.44) TP53ALOX15MEN1KMT2AALDH1A1
SCHEMBL12749081 0.85 TP53 (0.63) TP53ALOX15MEN1KMT2AKDM4E
SCHEMBL5929477 0.85 TP53 (0.52) TP53ALOX15MEN1KMT2AKDM4E
SCHEMBL1071885 0.81 TP53 (0.50) TP53ALOX15KDM4EMAPTALDH1A1
SCHEMBL974832 0.80 TP53 (0.46) TP53ALOX15KDM4EALDH1A1
SCHEMBL10676078 0.80 LSS (0.42) KDM4EMAPTDRD2DRD4
SCHEMBL15464534 0.79 TP53 (0.49) TP53ALOX15MEN1KMT2AKDM4E
SCHEMBL3242722 0.79 TP53 (0.49) TP53ALOX15MEN1KMT2AKDM4E
SCHEMBL6462571 0.79 TP53 (0.53) TP53ALOX15KDM4EMAPTALDH1A1
SCHEMBL3242725 0.79 TP53 (0.62) TP53ALOX15MEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009103022-A1 DERIVATIVES OF SUBSTITUTED FUSED RING CYCLOINDOLES AND METHODS OF THEIR USE ITHERX PHARMACEUTICALS, INC. (US) 2009-08-20 WO disclosed
WO-2009103022-A1 DERIVATIVES OF SUBSTITUTED FUSED RING CYCLOINDOLES AND METHODS OF THEIR USE ITHERX PHARMACEUTICALS, INC. (US) 2009-08-20 WO disclosed
EP-0393574-B1 Hexitol derivatives KYOWA HAKKO KOGYO KK (JP) 1996-01-31 EP disclosed
US-5053408-A Cardiovascular disorders KYOWA HAKKO KOGYO CO., LTD. (JP) 1991-10-01 US disclosed
EP-0393574-A2 Hexitol derivatives KYOWA HAKKO KOGYO CO., LTD. (JP) 1990-10-24 EP disclosed