SCHEMBL4028910

SCHEMBL4028910

COc1ccccc1CC[C@H]1NC(=O)CN[C@H]1c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 5/20 0.43
NR3C1 P04150 1/20 0.39
TAAR1 Q96RJ0 1/20 0.38
KDM1A O60341 2/20 0.38
MAOA P21397 2/20 0.38
MAOB P27338 1/20 0.38
ALDH1A1 P00352 1/20 0.38
SIGMAR1 Q99720 2/20 0.38
HRH3 Q9Y5N1 2/20 0.38
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4027969 1.00 TACR1 (0.43) TACR1NR3C1TAAR1KDM1AMAOA
Hydrochloric Acid SCHEMBL4026387 0.99 TACR1 (0.42) TACR1NR3C1TAAR1KDM1AMAOA
Hydrochloric Acid SCHEMBL4021093 0.99 TACR1 (0.42) TACR1NR3C1TAAR1KDM1AMAOA
SCHEMBL4026879 0.88 TACR1 (0.45) TACR1NR3C1KDM1AMAOAMAOB
SCHEMBL4027560 0.81 TACR1 (0.53) TACR1TAAR1KDM1AMAOAMAOB
Hydrochloric Acid SCHEMBL4020600 0.80 TACR1 (0.52) TACR1TAAR1KDM1AMAOAMAOB
Hydrochloric Acid SCHEMBL4029527 0.80 CHRNB4 (0.43) TACR1ALDH1A1
SCHEMBL17212309 0.71 TACR1 (0.62) TACR1SIGMAR1KCNH2
SCHEMBL9375929 0.70 TACR1 (0.58) TACR1KDM1AMAOAMAOB
SCHEMBL9375935 0.70 TACR1 (0.58) TACR1KDM1AMAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1338592-B1 Novel 2-phenylpiperazine derivatives NIPPON ZOKI PHARMACEUTICAL CO (JP) 2009-01-21 EP claimed