SCHEMBL4029185

SCHEMBL4029185

COC(=O)[C@]12CC[C@H](NCc3ccccc3)C[C@@H]1CCN(c1ccnc3ccc(OC)nc13)C2

nearest known ligand 0.45

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 9/20 0.44
CYP8B1 Q9UNU6 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3941340 0.81 KCNH2 (0.41) KCNH2
SCHEMBL3941342 0.81 KCNH2 (0.41) KCNH2
SCHEMBL4035891 0.81 KCNH2 (0.41) KCNH2
SCHEMBL4035886 0.81 KCNH2 (0.41) KCNH2
SCHEMBL3946267 0.77 KCNH2 (0.40) KCNH2CYP8B1
SCHEMBL3946262 0.77 KCNH2 (0.40) KCNH2CYP8B1
SCHEMBL3944928 0.77 CYP8B1 (0.37) KCNH2CYP8B1
SCHEMBL1224745 0.73 KCNH2 (0.38) KCNH2CYP8B1
SCHEMBL1224748 0.73 KCNH2 (0.38) KCNH2CYP8B1
SCHEMBL1223261 0.72 ALDH1A1 (0.45) KCNH2CYP8B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009034546-A2 TRANS-DECAHYDROISOQUINOLINE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2009-03-19 WO disclosed