SCHEMBL3944928

SCHEMBL3944928

COc1ccc2nccc(N3CC[C@H]4C[C@@H](NC(=O)OCc5ccccc5)CC[C@]4(CO)C3)c2n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP8B1 Q9UNU6 1/20 0.37
KCNH2 Q12809 7/20 0.37
SMPD3 Q9NY59 1/20 0.37
CPB1 P15086 1/20 0.35
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35
CTSK P43235 1/20 0.35
KDM1A O60341 1/20 0.35
MAOB P27338 1/20 0.35
ENPP2 Q13822 1/20 0.35
ATXN2 Q99700 1/20 0.35
DPP4 P27487 1/20 0.35
DPP7 Q9UHL4 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
ACHE P22303 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1223261 0.85 ALDH1A1 (0.45) CYP8B1KCNH2SMPD3CPB1CTSL
SCHEMBL1224380 0.81 ALDH1A1 (0.42) CYP8B1KCNH2SMPD3CPB1CTSL
SCHEMBL3942575 0.80 CYP8B1 (0.40) CYP8B1KCNH2
SCHEMBL4029185 0.77 KCNH2 (0.44) CYP8B1KCNH2
SCHEMBL4034084 0.75 KCNH2 (0.37) CYP8B1KCNH2
SCHEMBL3943077 0.75 KCNH2 (0.37) CYP8B1KCNH2
SCHEMBL4034087 0.75 KCNH2 (0.37) CYP8B1KCNH2
SCHEMBL3943081 0.75 KCNH2 (0.37) CYP8B1KCNH2
SCHEMBL3944808 0.72 HSD11B1 (0.45) KCNH2CTSLCTSBCTSKKDM1A
SCHEMBL1224645 0.72 KCNH2 (0.44) KCNH2SMPD3CTSLCTSBCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009034546-A2 TRANS-DECAHYDROISOQUINOLINE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2009-03-19 WO disclosed