SCHEMBL4029408

SCHEMBL4029408

CC(C)(C)OC(=O)NCCCOCCc1ccc(OCCN2CCSc3ccccc32)cc1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.52
LMNA P02545 1/20 0.52
MAPT P10636 1/20 0.52
KDM4E B2RXH2 1/20 0.47
MEN1 O00255 1/20 0.47
ALDH1A1 P00352 1/20 0.47
KMT2A Q03164 1/20 0.47
CA12 O43570 5/20 0.43
CA1 P00915 5/20 0.43
CA2 P00918 5/20 0.43
CA9 Q16790 5/20 0.43
SIGMAR1 Q99720 2/20 0.42
DRD2 P14416 4/20 0.41
POLB P06746 1/20 0.41
THRB P10828 1/20 0.41
RXFP1 Q9HBX9 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4032932 0.70 MAPT (0.51) TP53LMNAMAPTKDM4EMEN1
SCHEMBL4446760 0.70 MEN1 (0.55) MAPTMEN1KMT2ACA12CA1
SCHEMBL5101123 0.70 MAPT (0.53) TP53LMNAMAPTALDH1A1POLB
SCHEMBL23291147 0.69 LTA4H (0.53) KDM4ECA12CA1CA2CA9
SCHEMBL4656567 0.69 S1PR1 (0.60) CA12CA1CA2CA9SIGMAR1
SCHEMBL24920672 0.69 CA12 (0.67) MEN1KMT2ACA12CA1CA2
SCHEMBL5100503 0.69 LMNA (0.54) TP53LMNAMAPTPOLB
SCHEMBL13886735 0.69 NPC1 (0.57) MAPTMEN1KMT2ACA12CA1
SCHEMBL23291302 0.69 HRH3 (0.61) MAPTSIGMAR1POLB
SCHEMBL23291176 0.69 HRH3 (0.55) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569916-B1 SUBSTITUTED ARALKYL DERIVATIVES CADILA HEALTHCARE LTD (IN) 2009-01-07 EP claimed