SCHEMBL4030012

SCHEMBL4030012

Cc1cc(Cl)cnc1CN(Cc1ccc(C#N)cc1CO)CC(C)c1ccccn1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 1/20 0.35
KCNA5 P22460 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.31
AR P10275 4/20 0.31
FNTA P49354 2/20 0.30
FNTB P49356 2/20 0.30
PSEN1 P49768 1/20 0.30
PSEN2 P49810 1/20 0.30
APH1B Q8WW43 1/20 0.30
NCSTN Q92542 1/20 0.30
APH1A Q96BI3 1/20 0.30
PSENEN Q9NZ42 1/20 0.30
PGGT1B P53609 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4030008 0.81 CXCR4 (0.34) CXCR4ARPSEN1PSEN2APH1B
SCHEMBL4033761 0.78 CXCR4 (0.41) CXCR4SMN1; SMN2
SCHEMBL2085768 0.78 CNR1 (0.30) AR
SCHEMBL2084592 0.74 ADORA2A (0.37) CXCR4KCNA5
SCHEMBL2084581 0.74 CDK1 (0.35) AR
SCHEMBL2083828 0.70 CXCR4 (0.50) CXCR4
SCHEMBL4030664 0.68 PDE5A (0.35) CXCR4SMN1; SMN2FNTAFNTB
SCHEMBL25649146 0.67 MEN1 (0.35) KCNA5SMN1; SMN2FNTAFNTBPGGT1B
SCHEMBL4032125 0.65 CXCR4 (0.38) CXCR4SMN1; SMN2
SCHEMBL2084418 0.63 KDM4E (0.35) CXCR4AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613613-A4 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2009-03-25 EP disclosed
EP-1613613-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-01-11 EP disclosed
WO-2004091518-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2004-10-28 WO disclosed