SCHEMBL4030664

SCHEMBL4030664

COC(=O)c1cc(C#N)ccc1CN(Cc1ncc(Cl)cc1C)C(C)Cc1ccccn1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 4/20 0.35
EGLN1 Q9GZT9 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CXCR4 P61073 1/20 0.33
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
ALOX15 P16050 1/20 0.32
HSD17B10 Q99714 1/20 0.32
GRM4 Q14833 1/20 0.32
FNTA P49354 1/20 0.32
FNTB P49356 1/20 0.32
CNR1 P21554 1/20 0.32
CNR2 P34972 1/20 0.32
HPGD P15428 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
MRGPRX4 Q96LA9 1/20 0.32
MC4R P32245 1/20 0.32
PTGER4 P35408 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4030008 0.86 CXCR4 (0.34) PDE5AEGLN1CXCR4ALDH1A1CNR1
SCHEMBL4030668 0.82 CXCR4 (0.34) SMN1; SMN2CXCR4HCRTR1HCRTR2GRM4
SCHEMBL2080870 0.80 HPGD (0.33) PDE5AHCRTR1HCRTR2KDM4EALDH1A1
SCHEMBL2081315 0.77 CXCR4 (0.49) SMN1; SMN2CXCR4KDM4EALDH1A1HPGD
SCHEMBL4036473 0.74 KDM4E (0.41) EGLN1KDM4EALDH1A1ALOX15HSD17B10
SCHEMBL4033759 0.74 CXCR4 (0.39) CXCR4KDM4ENPSR1MC4R
SCHEMBL2084858 0.72 ADORA2A (0.40) HCRTR1HCRTR2KDM4EALDH1A1HPGD
SCHEMBL2082555 0.72 MRGPRX4 (0.39) PDE5ASMN1; SMN2KDM4EALDH1A1HPGD
SCHEMBL2084345 0.70 ADORA2A (0.36) KDM4EALDH1A1HPGDMRGPRX4
SCHEMBL4030012 0.68 CXCR4 (0.35) SMN1; SMN2CXCR4FNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613613-A4 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2009-03-25 EP disclosed
EP-1613613-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-01-11 EP disclosed
WO-2004091518-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2004-10-28 WO disclosed