SCHEMBL4030263

SCHEMBL4030263

Cc1cnc(CN(CCc2ccccn2)C2CCNCC2)c(C)c1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 10/20 0.46
SLC6A4 P31645 10/20 0.46
SLC6A3 Q01959 7/20 0.46
CXCR4 P61073 5/20 0.42
CYP2D6 P10635 4/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
RECQL P46063 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
CHRM2 P08172 1/20 0.37
CHRM4 P08173 1/20 0.37
CHRM5 P08912 1/20 0.37
CHRM1 P11229 1/20 0.37
CHRM3 P20309 1/20 0.37
KDM4E B2RXH2 2/20 0.36
POLB P06746 1/20 0.35
TSHR P16473 1/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4541280 0.82 CCR3 (0.45) CXCR4CYP2D6CYP2C9CYP2C19RECQL
SCHEMBL2082385 0.78 CXCR4 (0.42) SLC6A2SLC6A4SLC6A3CXCR4CYP2D6
SCHEMBL4039008 0.78 LMNA (0.47) POLB
SCHEMBL2082182 0.77 SLC6A2 (0.43) SLC6A2SLC6A4SLC6A3CXCR4CYP2D6
SCHEMBL2081862 0.77 SLC6A2 (0.39) SLC6A2SLC6A4SLC6A3CXCR4CYP2D6
SCHEMBL4030777 0.77 SLC6A2 (0.43) SLC6A2SLC6A4SLC6A3CXCR4CYP2D6
SCHEMBL4039684 0.75 CXCR4 (0.40) SLC6A2SLC6A4SLC6A3CXCR4CYP2D6
SCHEMBL2084715 0.75 CXCR4 (0.40) SLC6A2SLC6A4SLC6A3CXCR4CYP2D6
SCHEMBL2082739 0.75 CXCR4 (0.54) SLC6A2SLC6A4SLC6A3CXCR4CYP2D6
SCHEMBL2084727 0.74 CXCR4 (0.40) SLC6A2SLC6A4SLC6A3CXCR4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613613-A4 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2009-03-25 EP disclosed
EP-1613613-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-01-11 EP disclosed
WO-2004091518-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2004-10-28 WO disclosed