SCHEMBL4030469

SCHEMBL4030469

CNC(=O)c1[c]ccc2cc(C(O)(c3cn(C(c4ccccc4)(c4ccccc4)c4ccccc4)cn3)C(C)C)ccc12

nearest known ligand 0.37

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 7/20 0.37
CYP3A4 P08684 4/20 0.34
SIRT2 Q8IXJ6 10/20 0.33
RORC P51449 1/20 0.31
ACSS2 Q9NR19 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4023981 0.85 CYP17A1 (0.42) CYP17A1CYP3A4SIRT2ACSS2
SCHEMBL4029531 0.83 CYP17A1 (0.56) CYP17A1CYP3A4SIRT2RORCACSS2
SCHEMBL4027282 0.83 CYP17A1 (0.40) CYP17A1CYP3A4SIRT2RORC
SCHEMBL7266948 0.83 CYP17A1 (0.56) CYP17A1CYP3A4SIRT2RORCACSS2
SCHEMBL4031099 0.82 CYP17A1 (0.52) CYP17A1CYP3A4SIRT2ACSS2
SCHEMBL4027190 0.81 CYP3A4 (0.38) CYP17A1CYP3A4SIRT2
SCHEMBL4029977 0.79 CYP17A1 (0.55) CYP17A1CYP3A4SIRT2ACSS2
SCHEMBL4028814 0.78 CYP17A1 (0.36) CYP17A1CYP3A4SIRT2
SCHEMBL4031834 0.78 CYP17A1 (0.35) CYP17A1CYP3A4SIRT2
SCHEMBL5748871 0.78 CYP17A1 (0.53) CYP17A1CYP3A4SIRT2ACSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1222174-B1 IMIDAZOL-4-YLMETHANOLS USED AS INHIBITORS OF STEROID C17-20 LYASE TAKEDA PHARMACEUTICAL (JP) 2009-05-27 EP disclosed