SCHEMBL4036473

SCHEMBL4036473

COC(=O)c1cc(C#N)ccc1CN(CCc1ccccn1)Cc1ncccc1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 10/20 0.41
ALDH1A1 P00352 7/20 0.38
TDP1 Q9NUW8 2/20 0.38
HIF1A Q16665 1/20 0.36
MAPT P10636 2/20 0.36
LMNA P02545 1/20 0.36
PKM P14618 1/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
TSHR P16473 1/20 0.35
EGLN1 Q9GZT9 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
ALOX15 P16050 1/20 0.35
HSD17B10 Q99714 1/20 0.35
SCN9A Q15858 1/20 0.34
HPGD P15428 1/20 0.34
CRHBP P24387 1/20 0.34
CRHR2 Q13324 1/20 0.34
NPC1 O15118 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2084858 0.89 ADORA2A (0.40) KDM4EALDH1A1MAPTKMT2AADORA2A
SCHEMBL2082555 0.85 MRGPRX4 (0.39) KDM4EALDH1A1MAPTKMT2AADORA2A
SCHEMBL2084345 0.82 ADORA2A (0.36) KDM4EALDH1A1MEN1KMT2AADORA2A
SCHEMBL2081315 0.81 CXCR4 (0.49) KDM4EALDH1A1MAPTMEN1KMT2A
SCHEMBL2085274 0.78 ATR (0.36) KDM4EALDH1A1PKMKMT2AADORA2A
SCHEMBL4364791 0.78 F2 (0.40) KDM4EALDH1A1TDP1HIF1ATSHR
SCHEMBL4033882 0.76 KDM4E (0.33) KDM4EALDH1A1TDP1HIF1AMAPT
SCHEMBL22894683 0.75 TDP1 (0.53) KDM4ETDP1MAPTLMNAMEN1
SCHEMBL4030664 0.74 PDE5A (0.35) KDM4EALDH1A1EGLN1ALOX15HSD17B10
SCHEMBL4030668 0.73 CXCR4 (0.34) MEN1KMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613613-A4 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2009-03-25 EP disclosed
EP-1613613-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-01-11 EP disclosed
WO-2004091518-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2004-10-28 WO disclosed