SCHEMBL4031825

SCHEMBL4031825

Cc1ccc(-c2onc(C)c2N(C(=O)O)[C@H](C)c2ccccc2Br)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.38
RAB9A P51151 4/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
LPAR1 Q92633 3/20 0.36
LPAR3 Q9UBY5 2/20 0.36
TSHR P16473 3/20 0.36
ALOX15 P16050 1/20 0.36
ALDH1A1 P00352 3/20 0.35
NPSR1 Q6W5P4 2/20 0.35
HTT P42858 1/20 0.35
POLB P06746 2/20 0.35
IP6K1 Q92551 2/20 0.35
IP6K3 Q96PC2 2/20 0.35
IP6K2 Q9UHH9 2/20 0.35
LPAR2 Q9HBW0 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
NFKB1 P19838 2/20 0.34
NFKB2 Q00653 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4034111 0.87 BRD4 (0.37) NPC1RAB9AMEN1KMT2ALPAR1
SCHEMBL4034159 0.87 LPAR1 (0.44) NPC1RAB9AMEN1KMT2ALPAR1
SCHEMBL4034800 0.86 TRPV1 (0.38) LPAR1LPAR3NPSR1IP6K1IP6K3
SCHEMBL4028121 0.85 LPAR1 (0.44) NPC1RAB9AMEN1KMT2ALPAR1
SCHEMBL4030912 0.85 HDAC3 (0.40) LPAR1LPAR3TSHRNPSR1L3MBTL1
SCHEMBL4034108 0.81 LPAR1 (0.44) MEN1KMT2ALPAR1LPAR3ALDH1A1
SCHEMBL4028274 0.79 LPAR1 (0.37) NPC1MEN1KMT2ALPAR1LPAR3
SCHEMBL4032476 0.79 LPAR1 (0.43) MEN1KMT2ALPAR1LPAR3TSHR
SCHEMBL15437576 0.79 LPAR1 (0.43) MEN1KMT2ALPAR1LPAR3ALDH1A1
SCHEMBL4032913 0.77 LPAR1 (0.42) NPC1RAB9AMEN1KMT2ALPAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1258484-B1 NOVEL ISOXAZOLE AND THIAZOLE COMPOUNDS AND USE THEREOF AS DRUGS KYOWA HAKKO KIRIN CO LTD (JP) 2009-01-14 EP claimed