SCHEMBL4032258

SCHEMBL4032258

NS(=O)(=O)c1ccc(-n2nc(C(F)(F)F)c3c2CCCC3)cc1CO

nearest known ligand 0.55

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GRIA2 P42262 12/20 0.55
CYP1A2 P05177 3/20 0.55
CYP2D6 P10635 1/20 0.55
PTGS2 P35354 6/20 0.54
CYP2C19 P33261 1/20 0.53
CYP2C9 P11712 6/20 0.53
GAA P10253 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3109914 0.85 GRIA2 (0.60) GRIA2CYP1A2CYP2D6CYP2C19CYP2C9
SCHEMBL3104592 0.85 GRIA2 (0.63) GRIA2CYP1A2CYP2D6CYP2C19CYP2C9
SCHEMBL3103091 0.79 GRIA2 (0.53) GRIA2CYP1A2CYP2D6CYP2C19CYP2C9
SCHEMBL3107408 0.79 GRIA2 (0.77) GRIA2CYP1A2CYP2D6PTGS2CYP2C19
SCHEMBL8039330 0.79 PTGS2 (0.68) PTGS2
SCHEMBL8023227 0.77 PTGS2 (0.56) PTGS2
SCHEMBL8037470 0.77 PTGS2 (0.56) PTGS2
SCHEMBL3132184 0.77 GRIA2 (0.71) GRIA2CYP1A2CYP2D6CYP2C19CYP2C9
SCHEMBL4747751 0.73 GRIA2 (0.67) GRIA2CYP1A2CYP2D6CYP2C19CYP2C9
SCHEMBL8023576 0.73 PTGS2 (0.62) PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2051966-A2 HETEROCYCLES USEFUL AS INHIBITORS OF CARBONIC ANHYDRASE Pfizer Products Inc. (US) 2009-04-29 EP disclosed
WO-2008017932-A2 HETEROCYCLES USEFUL AS INHIBITORS OF CARBONIC ANHYDRASE PFIZER PRODUCTS INC. (US) 2008-02-14 WO disclosed