SCHEMBL4032356

SCHEMBL4032356

CC(C)Oc1ccc(I)cc1C(=O)NC(O)[C@H](C)c1c[nH]c2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.47
MEN1 O00255 3/20 0.47
CFTR P13569 3/20 0.38
NPC1 O15118 1/20 0.38
MAPT P10636 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
IGF1R P08069 1/20 0.36
MET P08581 1/20 0.36
SRC P12931 1/20 0.36
NR4A2 P43354 1/20 0.36
CREBBP Q92793 1/20 0.36
FFAR1 O14842 1/20 0.36
GPR84 Q9NQS5 1/20 0.36
PBRM1 Q86U86 1/20 0.36
LMNA P02545 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
TACR3 P29371 1/20 0.36
ITGB2 P05107 1/20 0.35
ICAM1 P05362 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4032359 1.00 KMT2A (0.47) KMT2AMEN1CFTRNPC1MAPT
SCHEMBL5149356 0.87 KDM4E (0.38) KMT2AMEN1CFTRMAPTFFAR1
SCHEMBL5149347 0.87 KDM4E (0.38) KMT2AMEN1CFTRMAPTFFAR1
SCHEMBL4038450 0.83 KMT2A (0.43) KMT2AMEN1CFTRNPC1MAPT
SCHEMBL4038446 0.83 KMT2A (0.43) KMT2AMEN1CFTRNPC1MAPT
SCHEMBL4035465 0.81 KMT2A (0.42) KMT2AMEN1NPC1MAPTNPSR1
SCHEMBL4035456 0.81 KMT2A (0.42) KMT2AMEN1NPC1MAPTNPSR1
SCHEMBL4032286 0.80 KMT2A (0.41) KMT2AMEN1NPC1MAPTNPSR1
SCHEMBL4032288 0.80 KMT2A (0.41) KMT2AMEN1NPC1MAPTNPSR1
SCHEMBL4037068 0.79 KMT2A (0.40) KMT2AMEN1MAPTNPSR1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2019102-A1 Alkylacetylene substituted Acyltryptophanols Bayer Schering Pharma AG (DE) 2009-01-28 EP disclosed