SCHEMBL4032452

SCHEMBL4032452

COC(=O)/C(=C\c1ccc2ccccc2c1)CC(=O)O

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.56
RECQL P46063 1/20 0.49
GLO1 Q04760 1/20 0.48
APP P05067 1/20 0.45
MAPT P10636 1/20 0.45
AKR1C3 P42330 1/20 0.45
PTPN7 P35236 1/20 0.42
DHODH Q02127 1/20 0.41
NQO2 P16083 1/20 0.41
PPARA Q07869 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4032454 1.00 PTGS2 (0.56) PTGS2RECQLGLO1APPMAPT
SCHEMBL11685334 0.84 PTGS2 (0.55) PTGS2APPMAPTAKR1C3NQO2
SCHEMBL28251651 0.84 PTGS2 (0.52) PTGS2APPMAPTAKR1C3
SCHEMBL1915834 0.83 RECQL (0.69) RECQLMAPTAKR1C3
SCHEMBL1915838 0.83 RECQL (0.69) RECQLMAPTAKR1C3
SCHEMBL1915837 0.83 RECQL (0.69) RECQLMAPTAKR1C3
SCHEMBL27725356 0.82 RECQL (0.58) PTGS2RECQL
SCHEMBL22231419 0.80 PTGS2 (0.49) PTGS2MAPT
SCHEMBL22231431 0.80 AKR1C3 (0.48) PTGS2GLO1APPMAPTAKR1C3
SCHEMBL22231429 0.80 AKR1C3 (0.48) PTGS2GLO1APPMAPTAKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1587795-B1 N- (1-BENZYL-2-OXO-2- (1-PIPERAZINYL) ETHYL) -1-PIPERIDINCARBOXAMID-DERIVATIVES AND RELATED COMPOUNDS USE AS CGRP-ANTAGONISTS FOR TREATING A HEADACHE BOEHRINGER INGELHEIM INT (DE) 2009-05-13 EP disclosed