SCHEMBL4032892

SCHEMBL4032892

CC(C)(C)OC(=O)NCCCn1c2c(c3cc(Br)ccc31)CCCC2

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.50
KRAS P01116 4/20 0.44
SCARB1 Q8WTV0 4/20 0.44
HSD17B10 Q99714 1/20 0.44
CAMK2D Q13557 1/20 0.43
HDAC1 Q13547 2/20 0.43
HDAC6 Q9UBN7 2/20 0.43
DYRK1A Q13627 1/20 0.42
ACLY P53396 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30981928 0.94 HSD17B10 (0.46) CNR2KRASSCARB1HSD17B10HDAC1
SCHEMBL30981996 0.92 KRAS (0.46) CNR2KRASSCARB1HSD17B10CAMK2D
SCHEMBL4024465 0.87 CNR2 (0.56) CNR2SCARB1HSD17B10DYRK1AACLY
SCHEMBL4023805 0.87 SCARB1 (0.61) CNR2SCARB1HSD17B10HDAC1HDAC6
SCHEMBL30981976 0.86 MTNR1A (0.44) CNR2KRASHSD17B10CAMK2DHDAC1
SCHEMBL15798202 0.81 CNR2 (0.67) CNR2CAMK2DHDAC1HDAC6DYRK1A
SCHEMBL30981883 0.79 KRAS (0.60) CNR2KRASHDAC1HDAC6
SCHEMBL15798230 0.79 DYRK1A (0.56) CNR2CAMK2DDYRK1A
SCHEMBL30981942 0.77 PTGDR2 (0.44) CNR2HSD17B10
SCHEMBL30981901 0.77 MTNR1A (0.39) CNR2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009103022-A1 DERIVATIVES OF SUBSTITUTED FUSED RING CYCLOINDOLES AND METHODS OF THEIR USE ITHERX PHARMACEUTICALS, INC. (US) 2009-08-20 WO disclosed