SCHEMBL4033752

SCHEMBL4033752

O=C(O)Oc1nc(-c2cccs2)n(CC(F)(F)F)c(=O)c1O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERCC1 P07992 2/20 0.43
FEN1 P39748 2/20 0.43
ERCC4 Q92889 2/20 0.43
ALDH1A1 P00352 8/20 0.39
KDM4E B2RXH2 5/20 0.39
HPGD P15428 4/20 0.38
POLB P06746 2/20 0.38
ELANE P08246 5/20 0.36
LMNA P02545 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
PLA2G1B P04054 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ATG4B Q9Y4P1 1/20 0.36
MAPK1 P28482 1/20 0.36
NPSR1 Q6W5P4 1/20 0.35
SMPD3 Q9NY59 1/20 0.35
HTT P42858 2/20 0.35
CYP1A2 P05177 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4025292 0.85 ERCC1 (0.48) ERCC1FEN1ERCC4ALDH1A1KDM4E
SCHEMBL4028670 0.83 ALDH1A1 (0.50) ERCC1FEN1ERCC4ALDH1A1KDM4E
SCHEMBL4029715 0.83 ERCC1 (0.63) ERCC1FEN1ERCC4ALDH1A1KDM4E
SCHEMBL4032043 0.79 ERCC1 (0.67) ERCC1FEN1ERCC4ALDH1A1KDM4E
SCHEMBL4029729 0.78 MAPT (0.47) ERCC1FEN1ERCC4ALDH1A1KDM4E
SCHEMBL4025290 0.68 ERCC1 (0.71) ERCC1FEN1ERCC4ALDH1A1KDM4E
SCHEMBL4028669 0.66 FEN1 (0.65) ERCC1FEN1ERCC4ALDH1A1KDM4E
SCHEMBL11858866 0.61 ALDH1A1 (0.39) ALDH1A1KDM4EHPGDPOLBLMNA
SCHEMBL11863646 0.61 ALDH1A1 (0.41) ALDH1A1KDM4EHPGDPOLBLMNA
SCHEMBL4027681 0.61 ERCC1 (0.41) ERCC1FEN1ERCC4ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3022199-A1 CYANOTRIAZOLE COMPOUNDS Otsuka Pharmaceutical Co., Ltd. (JP) 2016-05-25 EP claimed
WO-2015008872-A1 CYANOTRIAZOLE COMPOUNDS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2015-01-22 WO claimed
WO-2009016216-A1 TRIAZOLE DERIVATIVES AS SCD INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2009-02-05 WO claimed
CN-101918395-A Triazole oxadiazole derivatives MERCK SERONO SA 2010-12-15 CN disclosed
CN-101558066-A Pyrrole derivatives with antibacterial activity ASTRAZENECA AB (SE) 2009-10-14 CN disclosed
WO-2009016216-A1 TRIAZOLE DERIVATIVES AS SCD INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2009-02-05 WO disclosed
CN-100390169-C Hydroxymethyl substituted dihydroisoxazole derivatives useful as antibiotic agents ASTRAZENECA AB (SE) 2008-05-28 CN disclosed
CN-1753888-A Hydroxymethyl substituted dihydroisoxazole derivatives useful as antibiotic agents ASTRAZENECA AB (SE) 2006-03-29 CN disclosed
CN-1742015-A Oxazolidinone and / or isoxazoline derivatives as antibacterial agents ASTRAZENECA AB (SE) 2006-03-01 CN disclosed
CN-1227229-C Ethylene derivatives and pesticides containing the same NISSAN CHEMICAL IND LTD (JP) 2005-11-16 CN disclosed
CN-1216530-A Ethylene derivatives and pesticides containing the same NISSAN CHEMICAL IND LTD (JP) 1999-05-12 CN disclosed