SCHEMBL4033868

SCHEMBL4033868

CC(O)(c1ccc2c3c(ccc2c1)OCC3)c1c[nH]cn1

nearest known ligand 0.32

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 4/20 0.32
CYP2C8 P10632 1/20 0.32
KDM4E B2RXH2 1/20 0.31
NPC1 O15118 1/20 0.31
MAPT P10636 1/20 0.31
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4030416 0.94 CYP17A1 (0.31) CYP17A1CYP2C8
SCHEMBL4027318 0.87 MTNR1A (0.30)
SCHEMBL4027830 0.87 CYP17A1 (0.41) CYP17A1CYP2C8CYP3A4
SCHEMBL4028828 0.81 CYP17A1 (0.40) CYP17A1CYP2C8CYP3A4
SCHEMBL4034379 0.81 MTNR1A (0.30)
SCHEMBL1414829 0.74 CYP17A1 (0.58) CYP17A1CYP2C8CYP3A4
SCHEMBL4030413 0.72 NPC1 (0.32) NPC1MAPT
SCHEMBL5753491 0.70 CYP17A1 (0.47) CYP17A1KDM4ENPC1CYP3A4
SCHEMBL7266762 0.69 CYP17A1 (0.42) CYP17A1CYP3A4
SCHEMBL8128778 0.66 MAOA (0.44) KDM4ENPC1MAPTCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1222174-B1 IMIDAZOL-4-YLMETHANOLS USED AS INHIBITORS OF STEROID C17-20 LYASE TAKEDA PHARMACEUTICAL (JP) 2009-05-27 EP disclosed
US-6649643-B1 Antitumor, anticarcinogenic, and antimetastasis agents; benign prostatic hyperplasia, alopecia, endometriosis, uterine myoma, hirsutism, virilism, precocious puberty, mastopathy, and polycystic overay syndrome treatment TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-11-18 US disclosed
EP-1222174-A1 IMIDAZOL-4-YLMETHANOLS USED AS INHIBITORS OF STEROID C17-20 LYASE Takeda Chemical Industries, Ltd. (JP) 2002-07-17 EP disclosed
WO-2001030762-A1 IMIDAZOL-4-YLMETHANOLS USE AS INHIBITORS OF STEROID C17-20 LYASE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-03 WO disclosed