SCHEMBL4034696

SCHEMBL4034696

O=C1Cc2ccc(NC(=O)c3ccccc3NCc3ccc(C(=O)O)nc3)cc2N1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 1/20 0.47
IRAK4 Q9NWZ3 1/20 0.47
P4HTM Q9NXG6 1/20 0.42
KIT P10721 10/20 0.42
BRAF P15056 10/20 0.42
RXFP1 Q9HBX9 1/20 0.42
KMT2A Q03164 1/20 0.42
TRPV1 Q8NER1 2/20 0.42
FLT1 P17948 1/20 0.42
KDR P35968 1/20 0.42
SCD O00767 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4034859 0.93 IRAK4 (0.56) JAK3IRAK4P4HTMKITBRAF
SCHEMBL6542886 0.92 JAK3 (0.51) JAK3IRAK4KITBRAFTRPV1
SCHEMBL4034820 0.88 JAK3 (0.46) JAK3IRAK4KITBRAFRXFP1
SCHEMBL4042743 0.88 KIT (0.53) KITBRAF
SCHEMBL4034704 0.87 JAK3 (0.46) JAK3IRAK4KITBRAFRXFP1
SCHEMBL6542947 0.85 JAK3 (0.59) JAK3IRAK4KITBRAFFLT1
SCHEMBL4042030 0.84 JAK3 (0.47) JAK3IRAK4KITBRAFFLT1
SCHEMBL6792344 0.81 RXFP1 (0.42) JAK3IRAK4KITBRAFRXFP1
SCHEMBL4036359 0.81 JAK3 (0.54) JAK3IRAK4KITBRAFFLT1
SCHEMBL4032722 0.81 KIT (0.50) KITBRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1392680-B1 SELECTIVE ANTHRANILAMIDE PYRIDINE AMIDES AS INHIBITORS OF VEGFR-2 AND VEGFR-3 BAYER SCHERING PHARMA AG (DE) 2009-07-22 EP disclosed
US-20040254185-A1 Selective anthranilamide pyridine amides as inhibitors of vegfr-2 and vegfr-3 BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2004-12-16 US disclosed
EP-1392680-A2 SELECTIVE ANTHRANILAMIDE PYRIDINE AMIDES AS INHIBITORS OF VEGFR-2 AND VEGFR-3 SCHERING AKTIENGESELLSCHAFT (DE) 2004-03-03 EP disclosed
WO-2002090352-A2 SELECTIVE ANTHRANILAMIDE PYRIDINE AMIDES AS INHIBITORS OF VEGFR-2 AND VEGFR-3 SCHERING AKTIENGESELLSCHAFT (DE) 2002-11-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040254185-A1 Selective anthranilamide pyridine amides as inhibitors of vegfr-2 and vegfr-3 FLT4, KDR, FLT1 JAK3 33/4885IRAK4 159/4885P4HTM 441/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.