SCHEMBL4034774

SCHEMBL4034774

CC(CNC(=O)C1CN(C(=O)Nc2ccccc2-c2ccccc2)CCN1S(=O)(=O)c1cccc2cccnc12)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 4/20 0.52
ALDH1A1 P00352 3/20 0.46
HPGD P15428 1/20 0.46
TP53 P04637 1/20 0.44
THRB P10828 1/20 0.44
HCRTR1 O43613 1/20 0.43
KMT2A Q03164 1/20 0.43
POLB P06746 1/20 0.43
MAPT P10636 3/20 0.42
TSHR P16473 4/20 0.42
LMNA P02545 2/20 0.42
HSP90AA1 P07900 1/20 0.42
GFER P55789 1/20 0.42
FABP1 P07148 1/20 0.41
MAPK1 P28482 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4037109 0.85 GAA (0.57) GAAALDH1A1HPGDTP53THRB
SCHEMBL4033096 0.84 GAA (0.60) GAAALDH1A1HPGDTP53HCRTR1
SCHEMBL1382942 0.83 GAA (0.56) GAAALDH1A1HPGDTP53THRB
SCHEMBL4032554 0.82 QPCT (0.47) GAAALDH1A1HPGDTP53THRB
SCHEMBL4034972 0.82 QPCT (0.47) GAAALDH1A1HPGDTP53THRB
SCHEMBL4033581 0.82 GAA (0.57) GAAALDH1A1HPGDHCRTR1KMT2A
SCHEMBL4032274 0.79 GAA (0.55) GAAALDH1A1HPGDTP53THRB
SCHEMBL4210429 0.79 GAA (0.53) GAAALDH1A1HPGDTP53HCRTR1
SCHEMBL4032496 0.79 ALDH1A1 (0.51) GAAALDH1A1HPGDPOLBMAPT
Trifluoroacetic Acid SCHEMBL4034617 0.79 QPCT (0.44) GAAALDH1A1HPGDTP53THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1592389-B1 PIPERAZINE-2-CARBOXAMIDE DERIVATIVES SERONO LAB (CH) 2009-04-22 EP disclosed