SCHEMBL4035203

SCHEMBL4035203

CSCCC1NC2(CCN(OC(=O)O)CC2)NC1=O

nearest known ligand 0.37

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 2/20 0.37
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2941098 0.85 HDAC8 (0.34) HDAC8
SCHEMBL4037642 0.85 HDAC8 (0.34) HDAC8
SCHEMBL1802720 0.84 HDAC8 (0.40) HDAC8KDM4EALDH1A1MAPTTDP1
SCHEMBL3927548 0.84 HDAC8 (0.40) HDAC8KDM4EALDH1A1MAPTTDP1
SCHEMBL4033021 0.78 HDAC8 (0.34) HDAC8ALDH1A1MAPT
SCHEMBL2939814 0.77 HDAC8 (0.36) HDAC8
Hydrochloric Acid SCHEMBL1800200 0.76 HDAC8 (0.35) HDAC8
SCHEMBL4039483 0.73 CCR5 (0.34) HDAC8
SCHEMBL4035139 0.71 GAA (0.43) KDM4EALDH1A1MAPT
SCHEMBL1801346 0.71 HSD11B1 (0.43) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730144-B1 SUBSTITUTED 1,4,8-TRIAZASPIRO¬4.5 DECAN-2-ONE COMPOUNDS GRUENENTHAL GMBH (DE) 2009-06-10 EP disclosed