SCHEMBL4035596

SCHEMBL4035596

[CH2]N(C)CCc1c[nH]c2ccccc12

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 6/20 0.76
HTR1A P08908 5/20 0.76
HTR2C P28335 4/20 0.76
HTR2B P41595 3/20 0.76
HTR6 P50406 4/20 0.67
SLC6A4 P31645 2/20 0.67
ADRA2A P08913 2/20 0.61
ADRA2B P18089 2/20 0.61
ADRA2C P18825 2/20 0.61
ADRA1A P35348 2/20 0.61
HRH1 P35367 2/20 0.61
ADRA1B P35368 2/20 0.61
HTR1D P28221 2/20 0.61
SLC6A2 P23975 1/20 0.61
HTR1E P28566 1/20 0.61
DRD3 P35462 1/20 0.61
OPRK1 P41145 1/20 0.61
SLC6A3 Q01959 1/20 0.61
SIGMAR1 Q99720 1/20 0.61
CYP3A4 P08684 3/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30896267 0.86 HTR2A (0.81) HTR2AHTR1AHTR2CHTR2BHTR6
N,N-Dimethyltryptamine SCHEMBL29350959 0.86 HTR2A (1.00) HTR2AHTR1AHTR2CHTR2BHTR6
N,N-Dimethyltryptamine SCHEMBL27221709 0.86 HTR2A (1.00) HTR2AHTR1AHTR2CHTR2BHTR6
N,N-Dimethyltryptamine SCHEMBL335710 0.86 HTR2A (1.00) HTR2AHTR1AHTR2CHTR2BHTR6
N,N-Dimethyltryptamine SCHEMBL23069121 0.85 HTR2A (0.97) HTR2AHTR1AHTR2CHTR2BHTR6
N,N-Dimethyltryptamine SCHEMBL25285129 0.85 HTR2A (0.97) HTR2AHTR1AHTR2CHTR2BHTR6
SCHEMBL14950623 0.83 HTR1A (0.76) HTR2AHTR1AHTR2CHTR2BHTR6
SCHEMBL8861727 0.83 HTR2A (0.76) HTR2AHTR1AHTR2CHTR2BHTR6
SCHEMBL20970920 0.82 HTR1A (0.74) HTR2AHTR1AHTR2CHTR2BHTR6
SCHEMBL29504149 0.82 HTR1A (0.74) HTR2AHTR1AHTR2CHTR2BHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611088-B1 HYDROXAMATES AS THERAPEUTIC AGENTS PHARMACYCLICS INC (US) 2009-06-17 EP claimed
WO-2006069096-A1 SILANOL DERIVATIVES AS INHIBITORS OF HISTONE DEACETYLASE PHARMACYCLICS, INC. (US) 2006-06-29 WO disclosed