SCHEMBL4035867

SCHEMBL4035867

NC(=O)NC=O.O=C(c1ccccc1)N1CCN(S(=O)(=O)c2ccccc2)C(C(c2ccccc2)c2ccccc2)C1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA1 P00915 5/20 0.46
CA2 P00918 5/20 0.46
CA9 Q16790 5/20 0.46
CA4 P22748 4/20 0.46
MMP1 P03956 4/20 0.45
MMP9 P14780 4/20 0.45
MMP13 P45452 4/20 0.45
MMP3 P08254 2/20 0.45
MMP7 P09237 2/20 0.45
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
TSHR P16473 1/20 0.42
CYP2C19 P33261 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
CA12 O43570 1/20 0.39
CA7 P43166 1/20 0.39
CA14 Q9ULX7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4040817 0.85 MAOB (0.42) CA1CA2CA9CA4L3MBTL1
SCHEMBL4035295 0.68 MMP1 (0.60) CA1CA2CA9CA4MMP1
SCHEMBL6189627 0.68 MMP1 (0.52) CA1CA2CA9CA4MMP1
SCHEMBL10681034 0.67 CA1 (0.54) CA1CA2CA9CA4MMP1
SCHEMBL5654242 0.65 MMP1 (0.56) CA1CA2CA9CA4MMP1
SCHEMBL6189161 0.65 CACNA2D1 (0.49) MMP1MMP9MMP13MMP3MMP7
SCHEMBL14393122 0.65 MMP1 (0.53) CA1CA2CA9CA4MMP1
SCHEMBL5324061 0.64 MMP1 (0.58) CA1CA2CA9CA4MMP1
SCHEMBL5324461 0.64 MMP1 (0.55) CA1CA2CA9CA4MMP1
SCHEMBL3715208 0.64 MMP1 (0.55) CA1CA2CA9CA4MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1592389-B1 PIPERAZINE-2-CARBOXAMIDE DERIVATIVES SERONO LAB (CH) 2009-04-22 EP claimed