SCHEMBL6189161

SCHEMBL6189161

NC(=O)C1CN(C(=O)NC(c2ccccc2)c2ccccc2)CCN1S(=O)(=O)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 3/20 0.49
CACNA1B Q00975 3/20 0.49
CACNB1 Q02641 3/20 0.49
CACNA1C Q13936 2/20 0.49
LMNA P02545 1/20 0.47
MAPT P10636 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
MMP1 P03956 2/20 0.47
MMP9 P14780 2/20 0.47
MMP13 P45452 2/20 0.47
ALDH1A1 P00352 4/20 0.47
HTT P42858 1/20 0.46
USP2 O75604 1/20 0.46
MMP3 P08254 1/20 0.43
MMP7 P09237 1/20 0.43
GAA P10253 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1383367 0.81 GAA (0.58) LMNAMAPTALDH1A1HTTUSP2
SCHEMBL4041221 0.80 ALDH1A1 (0.49) LMNAMAPTNPSR1MMP1MMP9
SCHEMBL7346677 0.79 MMP1 (0.54) MMP1MMP9MMP13ALDH1A1MMP3
SCHEMBL1380921 0.76 MMP1 (0.54) LMNAMAPTMMP1MMP9MMP13
SCHEMBL6190434 0.75 GAA (0.48) LMNANPSR1ALDH1A1HTTUSP2
SCHEMBL17512449 0.74 CACNA2D1 (0.81) CACNA2D1CACNA1BCACNB1CACNA1CLMNA
SCHEMBL5234080 0.74 ALDH1A1 (0.53) MMP1MMP9MMP13ALDH1A1HTT
SCHEMBL1382978 0.73 SMN1; SMN2 (0.53) LMNAMMP1MMP9MMP13ALDH1A1
SCHEMBL1380848 0.72 CACNA2D1 (0.51) CACNA2D1CACNA1BCACNB1CACNA1CLMNA
SCHEMBL695071 0.72 MMP2 (0.59) LMNAMAPTNPSR1MMP9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1592389-A2 PIPERAZINE-2-CARBOXAMIDE DERIVATIVES Applied Research Systems ARS Holding N.V. (AN) 2005-11-09 EP disclosed
WO-2004071390-A2 PIPERAZINE-2-CARBOXAMIDE DERIVATIVES APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2004-08-26 WO disclosed