SCHEMBL4035990

SCHEMBL4035990

CCN(CCCCNC(=O)OC(C)(C)C)c1ncccc1C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.47
KDM4E B2RXH2 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CA12 O43570 4/20 0.41
CA1 P00915 4/20 0.41
CA2 P00918 4/20 0.41
CA9 Q16790 4/20 0.41
HDAC6 Q9UBN7 2/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
STING1 Q86WV6 1/20 0.41
CKS1B P61024 1/20 0.39
SKP1 P63208 1/20 0.39
SKP2 Q13309 1/20 0.39
CXCR4 P61073 1/20 0.39
BRD4 O60885 2/20 0.39
PDPK1 O15530 1/20 0.39
CCNB2 O95067 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4036156 0.82 CKS1B (0.45) CYP3A4KDM4EL3MBTL1TDP1CA12
SCHEMBL4036322 0.79 CKS1B (0.46) CYP3A4KDM4EL3MBTL1TDP1CA12
SCHEMBL4038789 0.78 DYRK1A (0.43) CYP3A4KDM4EL3MBTL1TDP1CA12
SCHEMBL4030707 0.78 CYP3A4 (0.46) CYP3A4KDM4EL3MBTL1TDP1CA12
SCHEMBL4039822 0.77 CKS1B (0.42) CYP3A4KDM4ETDP1CA12CA1
SCHEMBL2083428 0.76 CYP3A4 (0.43) CYP3A4KDM4EL3MBTL1TDP1CA12
SCHEMBL4035432 0.76 L3MBTL1 (0.48) CYP3A4L3MBTL1TDP1CA12CA1
SCHEMBL2081506 0.75 CYP3A4 (0.50) CYP3A4KDM4EL3MBTL1TDP1CA12
SCHEMBL4035993 0.74 CYP3A4 (0.47) CYP3A4KDM4EL3MBTL1TDP1CA12
SCHEMBL8747512 0.74 KMT2A (0.50) KDM4ETDP1CKS1BSKP1SKP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613613-A4 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2009-03-25 EP disclosed
EP-1613613-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-01-11 EP disclosed
WO-2004091518-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2004-10-28 WO disclosed