SCHEMBL4036156

SCHEMBL4036156

CCN(CCCCNC(=O)OC(C)(C)C)c1ccccn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CKS1B P61024 1/20 0.45
SKP1 P63208 1/20 0.45
SKP2 Q13309 1/20 0.45
CYP3A4 P08684 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
CA12 O43570 4/20 0.42
CA1 P00915 4/20 0.42
CA2 P00918 4/20 0.42
CA9 Q16790 4/20 0.42
SSTR4 P31391 1/20 0.41
DRD2 P14416 3/20 0.41
KDM4E B2RXH2 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
BRD4 O60885 1/20 0.40
LMNA P02545 1/20 0.40
PDPK1 O15530 1/20 0.40
CCNB2 O95067 1/20 0.40
PRKCB P05771 1/20 0.40
CDK1 P06493 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4036322 0.97 CKS1B (0.46) CKS1BSKP1SKP2CYP3A4TDP1
SCHEMBL4038789 0.84 DYRK1A (0.43) CKS1BSKP1SKP2CYP3A4TDP1
SCHEMBL4030707 0.84 CYP3A4 (0.46) CKS1BSKP1SKP2CYP3A4TDP1
SCHEMBL4039822 0.83 CKS1B (0.42) CKS1BSKP1SKP2CYP3A4TDP1
SCHEMBL4035990 0.82 CYP3A4 (0.47) CKS1BSKP1SKP2CYP3A4TDP1
SCHEMBL837529 0.80 CKS1B (0.64) CKS1BSKP1SKP2CYP3A4TDP1
SCHEMBL8747512 0.78 KMT2A (0.50) CKS1BSKP1SKP2TDP1KDM4E
SCHEMBL2840695 0.77 TDP1 (0.47) CKS1BSKP1SKP2CYP3A4TDP1
SCHEMBL4035432 0.77 L3MBTL1 (0.48) CYP3A4TDP1CA12CA1CA2
SCHEMBL3974693 0.77 TDP1 (0.47) CKS1BSKP1SKP2CYP3A4TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613613-A4 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2009-03-25 EP disclosed
EP-1613613-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-01-11 EP disclosed
WO-2004091518-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2004-10-28 WO disclosed