SCHEMBL4033882

SCHEMBL4033882

COC(=O)c1cc(C#N)ccc1CN(CCc1ccccn1)CC1(C(=O)OC(C)(C)C)Nc2ccccc2N1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.33
ALDH1A1 P00352 6/20 0.33
TDP1 Q9NUW8 1/20 0.33
ALOX15 P16050 1/20 0.32
HSD17B10 Q99714 1/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
PKM P14618 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
TSHR P16473 1/20 0.32
CYP1A2 P05177 1/20 0.31
SCN9A Q15858 1/20 0.30
MAPKAPK2 P49137 1/20 0.30
FNTA P49354 1/20 0.30
FNTB P49356 1/20 0.30
HIF1A Q16665 1/20 0.30
CXCR3 P49682 1/20 0.30
HCRTR1 O43613 1/20 0.30
HCRTR2 O43614 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7147425 0.77 CXCR4 (0.44)
SCHEMBL4036473 0.76 KDM4E (0.41) KDM4EALDH1A1TDP1ALOX15HSD17B10
SCHEMBL2084858 0.68 ADORA2A (0.40) KDM4EALDH1A1MAPTKMT2ACYP1A2
SCHEMBL2085274 0.68 ATR (0.36) KDM4EALDH1A1HSD17B10PKMKMT2A
SCHEMBL7149584 0.66 CXCR4 (0.40)
SCHEMBL2082555 0.65 MRGPRX4 (0.39) KDM4EALDH1A1MAPTKMT2A
SCHEMBL29575263 0.64 ALDH1A1 (0.52) KDM4EALDH1A1TDP1ALOX15HSD17B10
SCHEMBL2081315 0.64 CXCR4 (0.49) KDM4EALDH1A1MAPTMEN1KMT2A
SCHEMBL2084345 0.63 ADORA2A (0.36) KDM4EALDH1A1MEN1KMT2A
SCHEMBL4035655 0.63 DRD2 (0.39) KDM4EALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613613-A4 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2009-03-25 EP disclosed
EP-1613613-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-01-11 EP disclosed
WO-2004091518-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2004-10-28 WO disclosed