SCHEMBL4037144

SCHEMBL4037144

C#CCN1C(=O)C(CC(C)C)NC12CCN(SC(=O)O)CC2

nearest known ligand 0.33

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 7/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4032461 0.87 CCR5 (0.32) CCR5
SCHEMBL3925985 0.83 CCR5 (0.34) CCR5
SCHEMBL1800874 0.78 CCR5 (0.32) CCR5
SCHEMBL4035595 0.77 CCR5 (0.38) CCR5
SCHEMBL2999337 0.75
SCHEMBL1800729 0.75 CYP2D6 (0.50)
SCHEMBL3927335 0.73 POLB (0.39)
SCHEMBL1801638 0.73 CRBN (0.46)
SCHEMBL1802377 0.73 SMN1; SMN2 (0.45)
SCHEMBL1800759 0.72 HRH3 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730144-B1 SUBSTITUTED 1,4,8-TRIAZASPIRO¬4.5 DECAN-2-ONE COMPOUNDS GRUENENTHAL GMBH (DE) 2009-06-10 EP claimed