SCHEMBL4035595

SCHEMBL4035595

CC(C)CC1NC2(CCN(SC(=O)O)CC2)N(Cc2ccccc2C#N)C1=O

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 13/20 0.38
TSHR P16473 1/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
TACR1 P25103 2/20 0.34
FEN1 P39748 1/20 0.34
DPP4 P27487 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRL1 P41146 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4038035 0.89 CCR5 (0.36) CCR5TSHRSLC6A2SLC6A4TACR1
SCHEMBL3917088 0.88 CCR5 (0.39) CCR5TSHRSLC6A2SLC6A4TACR1
SCHEMBL4042715 0.87 FEN1 (0.33) TSHRFEN1DPP4OPRM1OPRL1
SCHEMBL4041157 0.86 CCR5 (0.38) CCR5SLC6A2SLC6A4DPP4OPRM1
SCHEMBL3922909 0.86 CCR5 (0.39) CCR5TSHRTACR1DPP4OPRM1
SCHEMBL4036456 0.83 CCR5 (0.36) CCR5DPP4
SCHEMBL1796739 0.83 CYP2D6 (0.40) CCR5TSHR
SCHEMBL3916341 0.80 POLB (0.40) CCR5DPP4
SCHEMBL1799349 0.78 MAPT (0.41) CCR5DPP4
SCHEMBL4037144 0.77 CCR5 (0.33) CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730144-B1 SUBSTITUTED 1,4,8-TRIAZASPIRO¬4.5 DECAN-2-ONE COMPOUNDS GRUENENTHAL GMBH (DE) 2009-06-10 EP claimed