SCHEMBL4038037

SCHEMBL4038037

CSCCC1NC2(CCN(C(=S)NC(=O)O)CC2)N(Cc2cccc(C#N)c2)C1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 2/20 0.37
FAAH O00519 1/20 0.37
DRD4 P21917 2/20 0.36
CHRM4 P08173 4/20 0.35
CCR3 P51677 1/20 0.34
CHRM2 P08172 2/20 0.34
CHRM1 P11229 2/20 0.34
GAA P10253 1/20 0.34
KMT2A Q03164 1/20 0.34
DRD3 P35462 1/20 0.34
CCR5 P51681 1/20 0.33
KCNH2 Q12809 1/20 0.33
DCUN1D1 Q96GG9 1/20 0.33
NTRK1 P04629 1/20 0.33
MLNR O43193 1/20 0.33
BRD4 O60885 1/20 0.33
JAK2 O60674 1/20 0.32
JAK1 P23458 1/20 0.32
TYK2 P29597 1/20 0.32
JAK3 P52333 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3914895 0.90 CHRM3 (0.40) CHRM3FAAHDRD4CHRM4CCR3
SCHEMBL3925657 0.90 CHRM3 (0.40) CHRM3FAAHDRD4CHRM4CCR3
SCHEMBL3925615 0.87 KDM4E (0.37) CHRM3FAAHDRD4CHRM4CHRM2
SCHEMBL3916929 0.87 CHRM3 (0.36) CHRM3FAAHDRD4CHRM4CCR3
SCHEMBL3925417 0.86 MEN1 (0.41) CHRM3CHRM4KMT2A
SCHEMBL1800614 0.86 RORC (0.40) CHRM3FAAHDRD4CHRM4CCR3
SCHEMBL4040064 0.85 CHRM3 (0.39) CHRM3FAAHDRD4CHRM4CCR3
SCHEMBL4038594 0.84 P2RX7 (0.33) CHRM4CHRM1GAAKMT2ACCR5
SCHEMBL1799605 0.84 MAPK1 (0.46) CHRM3FAAHMLNR
SCHEMBL4037652 0.84 CHRM3 (0.41) CHRM3FAAHDRD4CHRM4CCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730144-B1 SUBSTITUTED 1,4,8-TRIAZASPIRO¬4.5 DECAN-2-ONE COMPOUNDS GRUENENTHAL GMBH (DE) 2009-06-10 EP claimed