SCHEMBL4038499

SCHEMBL4038499

CC(C)CC(NC(=O)c1ccc(OC(F)F)cc1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)c1ccc[n+]([O-])c1

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSK P43235 12/20 0.50
CTSS P25774 3/20 0.39
POLB P06746 1/20 0.35
CCR1 P32246 1/20 0.35
CA2 P00918 2/20 0.35
CA1 P00915 1/20 0.35
CTSV O60911 2/20 0.34
CTSL P07711 2/20 0.34
IDO1 P14902 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4043807 0.92 CTSK (0.41) CTSKCTSSCCR1CTSVCTSL
SCHEMBL4042967 0.92 CTSK (0.52) CTSKCTSSPOLBCA2CTSL
SCHEMBL4045094 0.91 CTSK (0.51) CTSKCTSSPOLBCCR1CA2
SCHEMBL4039563 0.91 CTSK (0.54) CTSKCTSSCCR1CA2CA1
SCHEMBL4038667 0.90 CTSK (0.54) CTSKCTSSCCR1CA2CA1
SCHEMBL4045969 0.89 CTSK (0.56) CTSKCTSSCCR1CA2CA1
SCHEMBL4042980 0.89 CTSK (0.53) CTSKCTSSCCR1CA2CA1
SCHEMBL4039332 0.89 CTSK (0.53) CTSKCTSSPOLBCCR1CA2
SCHEMBL4040927 0.89 CTSK (0.51) CTSKCTSSPOLBCCR1CTSV
SCHEMBL4040650 0.88 CTSK (0.65) CTSKCTSSCCR1CA2CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed
EP-1678157-A4 HETEROCYCLIC COMPOUNDS AND METHODS OF MAKING AND USING THEREOF REDDY US THERAPEUTICS INC (US) 2009-03-18 EP disclosed
EP-1678157-A2 HETEROCYCLIC COMPOUNDS AND METHODS OF MAKING AND USING THEREOF Reddy US Therapeutics, Inc. (US) 2006-07-12 EP disclosed
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP disclosed
WO-2005042712-A2 HETEROCYCLIC COMPOUNDS AND METHODS OF MAKING AND USING THEREOF REDDY US THERAPEUTICS, INC. (US) 2005-05-12 WO disclosed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO disclosed