SCHEMBL4038718

SCHEMBL4038718

COC(=O)C=Cc1cc2c(s1)-c1cc(F)ccc1Oc1ccccc1-2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.40
ALDH1A1 P00352 4/20 0.40
GAA P10253 4/20 0.40
ESR1 P03372 4/20 0.36
L3MBTL1 Q9Y468 3/20 0.35
PRKDC P78527 1/20 0.34
NOTUM Q6P988 1/20 0.33
ALOX5 P09917 1/20 0.33
GLA P06280 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
CASP1 P29466 1/20 0.33
CASP7 P55210 1/20 0.33
ATM Q13315 1/20 0.33
HSD17B10 Q99714 1/20 0.33
KMT2A Q03164 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
P2RX4 Q99571 1/20 0.32
NR1H4 Q96RI1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4046001 1.00 KDM4E (0.40) KDM4EALDH1A1GAAESR1L3MBTL1
SCHEMBL6333988 0.90 KDM4E (0.39) KDM4EALDH1A1GAAESR1L3MBTL1
SCHEMBL4037837 0.88 GAA (0.39) KDM4EALDH1A1GAAESR1L3MBTL1
SCHEMBL4037833 0.88 GAA (0.39) KDM4EALDH1A1GAAESR1L3MBTL1
SCHEMBL4043399 0.87 HRH4 (0.38) KDM4EALDH1A1MAPK1KMT2ASMN1; SMN2
SCHEMBL4037785 0.87 HRH4 (0.38) KDM4EALDH1A1MAPK1KMT2ASMN1; SMN2
SCHEMBL4035860 0.87 ALOX5 (0.39) KDM4EALDH1A1GAAESR1L3MBTL1
SCHEMBL4035859 0.87 ALOX5 (0.39) KDM4EALDH1A1GAAESR1L3MBTL1
SCHEMBL4036046 0.75 HRH4 (0.39) KDM4EALDH1A1NOTUMTSHRMAPK1
SCHEMBL4036049 0.75 HRH4 (0.39) KDM4EALDH1A1NOTUMTSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1284977-B1 THIENODIBENZOAZULENE COMPOUNDS AS TUMOR NECROSIS FACTOR INHIBITORS GLAXOSMITHKLINE ZAGREB (HR) 2009-06-24 EP claimed
EP-1284977-B1 THIENODIBENZOAZULENE COMPOUNDS AS TUMOR NECROSIS FACTOR INHIBITORS GLAXOSMITHKLINE ZAGREB (HR) 2009-06-24 EP disclosed