SCHEMBL4039419

SCHEMBL4039419

O=C(NC1(C(=O)N2CCC3C2C(=O)CN3C(=O)Cc2ccccn2)CCCCC1)c1ccc(-c2cccs2)cc1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 7/20 0.39
DPP4 P27487 1/20 0.38
PREP P48147 1/20 0.38
HDAC2 Q92769 3/20 0.35
DRD4 P21917 6/20 0.35
DRD2 P14416 5/20 0.35
HTR2A P28223 3/20 0.35
CHRM4 P08173 1/20 0.34
KCNH2 Q12809 2/20 0.34
TACR3 P29371 1/20 0.34
HDAC3 O15379 1/20 0.33
CTSL P07711 1/20 0.33
CTSB P07858 1/20 0.33
CTSS P25774 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
CTSK P43235 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4040806 0.88 CTSK (0.38) HDAC1DPP4PREPHDAC2DRD4
SCHEMBL4043068 0.87 HDAC1 (0.36) HDAC1DPP4PREPHDAC2DRD4
SCHEMBL4048563 0.87 HDAC1 (0.40) HDAC1DPP4PREPHDAC2DRD4
SCHEMBL4043621 0.84 CTSK (0.39) HDAC1DPP4PREPDRD4DRD2
SCHEMBL4042382 0.82 HDAC1 (0.35) HDAC1DPP4PREPHDAC2DRD4
SCHEMBL4039472 0.78 HDAC1 (0.35) HDAC1DPP4PREPHDAC2CHRM4
SCHEMBL4040909 0.77 GPR132 (0.36) HDAC1DPP4PREPHDAC2DRD4
SCHEMBL4039814 0.76 HDAC1 (0.36) HDAC1DPP4PREPHDAC2DRD4
SCHEMBL6209625 0.76 HDAC1 (0.35) HDAC1DPP4PREPDRD4DRD2
SCHEMBL4043991 0.76 HDAC1 (0.35) HDAC1DPP4PREPDRD4DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed