SCHEMBL4039677

SCHEMBL4039677

CNCCOc1ccc(C(=O)NO)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.58
PLK1 P53350 2/20 0.57
CA1 P00915 1/20 0.56
CA2 P00918 1/20 0.56
HDAC6 Q9UBN7 3/20 0.53
KDM1A O60341 2/20 0.53
HTR1D P28221 1/20 0.53
HTR1B P28222 1/20 0.53
MMP1 P03956 1/20 0.52
HDAC2 Q92769 1/20 0.52
HDAC8 Q9BY41 1/20 0.52
KDM4E B2RXH2 1/20 0.50
MEN1 O00255 1/20 0.50
ALDH1A1 P00352 1/20 0.50
HTT P42858 1/20 0.50
KMT2A Q03164 1/20 0.50
MAPT P10636 1/20 0.50
USP2 O75604 1/20 0.50
ALOX15 P16050 1/20 0.50
TSHR P16473 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9629138 0.88 PLK1 (0.73) NPC1PLK1HTR1DHTR1BKDM4E
SCHEMBL25581165 0.84 NPC1 (0.55) NPC1PLK1CA1CA2HTR1D
SCHEMBL6671125 0.83 MMP1 (0.72) PLK1HDAC6MMP1KDM4ETSHR
SCHEMBL10065842 0.83 TSHR (0.71) NPC1HTR1DHTR1BKDM4EALDH1A1
SCHEMBL14880162 0.83 PLK1 (0.75) NPC1PLK1CA1CA2MMP1
SCHEMBL5141541 0.83 L3MBTL1 (0.70) NPC1PLK1HTR1DHTR1BKDM4E
SCHEMBL24600195 0.83 NPC1 (0.66) NPC1PLK1MMP1KDM4EMEN1
SCHEMBL12966671 0.83 NPC1 (0.54) NPC1PLK1HTR1DHTR1BKDM4E
SCHEMBL5051932 0.82 GAA (0.61) PLK1CA1CA2HDAC6KDM1A
SCHEMBL13715503 0.81 PARP10 (0.62) NPC1PLK1CA1CA2HTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611088-B1 HYDROXAMATES AS THERAPEUTIC AGENTS PHARMACYCLICS INC (US) 2009-06-17 EP claimed