SCHEMBL4040292

SCHEMBL4040292

CN(C)CCCOCc1cc2c(s1)-c1ccc(Br)cc1Sc1ccccc1-2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.38
MEN1 O00255 2/20 0.38
CYP1A2 P05177 3/20 0.36
CYP2D6 P10635 3/20 0.36
CYP2C19 P33261 3/20 0.36
CYP3A4 P08684 3/20 0.36
MTOR P42345 2/20 0.36
TP53 P04637 2/20 0.36
THPO P40225 2/20 0.36
NFKB1 P19838 1/20 0.36
MAPK1 P28482 1/20 0.36
LMNA P02545 4/20 0.35
PMP22 Q01453 2/20 0.35
GMNN O75496 1/20 0.35
CHRM2 P08172 4/20 0.32
HTR1A P08908 4/20 0.32
ADRA2A P08913 4/20 0.32
CHRM1 P11229 4/20 0.32
DRD1 P21728 4/20 0.32
SLC6A2 P23975 4/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4042137 0.99 KMT2A (0.40) KMT2AMEN1CYP1A2CYP2D6CYP2C19
SCHEMBL4040864 0.94 CYP3A4 (0.37) KMT2AMEN1CYP1A2CYP2D6CYP2C19
Hydrochloric Acid SCHEMBL4042271 0.93 LMNA (0.38) KMT2AMEN1CYP1A2CYP2D6CYP2C19
SCHEMBL4043965 0.93 KMT2A (0.35) KMT2AMEN1CYP1A2CYP2D6CYP2C19
Hydrochloric Acid SCHEMBL4037158 0.92 KMT2A (0.36) KMT2AMEN1CYP1A2CYP2D6CYP2C19
SCHEMBL4039594 0.92 MEN1 (0.39) KMT2AMEN1CYP1A2CYP2D6CYP2C19
Hydrochloric Acid SCHEMBL4037809 0.90 KMT2A (0.40) KMT2AMEN1CYP1A2CYP2D6CYP2C19
SCHEMBL6333770 0.89 KMT2A (0.39) KMT2AMEN1CYP1A2CYP2D6CYP2C19
SCHEMBL6335341 0.88 CYP3A4 (0.50) KMT2AMEN1CYP1A2CYP2D6CYP2C19
SCHEMBL4041467 0.88 CYP3A4 (0.50) KMT2AMEN1CYP1A2CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1284977-B1 THIENODIBENZOAZULENE COMPOUNDS AS TUMOR NECROSIS FACTOR INHIBITORS GLAXOSMITHKLINE ZAGREB (HR) 2009-06-24 EP claimed